SCHEMBL8254

SCHEMBL8254

O=c1c(-c2ccccc2)c(CN2CCOCC2)oc2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.56
RAB9A P51151 3/20 0.56
ATM Q13315 1/20 0.56
ALDH1A1 P00352 7/20 0.51
HSD17B10 Q99714 5/20 0.51
KDM4E B2RXH2 4/20 0.51
HPGD P15428 2/20 0.51
RCE1 Q9Y256 1/20 0.51
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
MAPT P10636 4/20 0.47
NPSR1 Q6W5P4 2/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
KCNA3 P22001 1/20 0.46
GAA P10253 2/20 0.44
ALOX15 P16050 2/20 0.44
TSHR P16473 2/20 0.44
MAOB P27338 1/20 0.44
KLK7 P49862 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9032 0.99 NPC1 (0.55) NPC1RAB9AATMALDH1A1HSD17B10
SCHEMBL30680218 0.91 NPC1 (0.56) NPC1RAB9AATMALDH1A1HSD17B10
SCHEMBL7856 0.91 NPC1 (0.56) NPC1RAB9AATMALDH1A1HSD17B10
Hydrochloric Acid SCHEMBL9337 0.90 NPC1 (0.55) NPC1RAB9AATMALDH1A1HSD17B10
Hydrochloric Acid SCHEMBL29651829 0.90 NPC1 (0.55) NPC1RAB9AATMALDH1A1HSD17B10
SCHEMBL1443636 0.86 CA1 (0.48) NPC1RAB9AATMALDH1A1HSD17B10
SCHEMBL8381 0.86 ALDH1A1 (0.57) NPC1RAB9AATMALDH1A1HSD17B10
Hydrochloric Acid SCHEMBL8872 0.85 ALDH1A1 (0.56) NPC1RAB9AATMALDH1A1HSD17B10
SCHEMBL6667780 0.78 NPC1 (0.51) NPC1RAB9AATMALDH1A1HSD17B10
SCHEMBL9656 0.76 GABRP (0.46) NPC1RAB9AATMALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 61 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240360095-A1 NOVEL KINASE MODULATORS RHIZEN PHARMACEUTICALS AG (CH) 2024-10-31 US claimed
US-11858907-B2 Kinase modulators RHIZEN PHARMACEUTICALS AG (CH) 2024-01-02 US claimed
EP-4292596-A1 METHOD AND COMBINATION FOR TREATING TUMORS Curon Biopharmaceutical (Shanghai) Co., Limited (CN) 2023-12-20 EP claimed
US-20200239427-A1 NOVEL KINASE MODULATORS RHIZEN PHARMACEUTICALS AG (CH) 2020-07-30 US claimed
EP-3050876-A2 KINASE MODULATORS Rhizen Pharmaceuticals S.A. (CH) 2016-08-03 EP claimed
EP-2496567-A2 NOVEL BENZOPYRAN KINASE MODULATORS Rhizen Pharmaceuticals S.A. (CH) 2012-09-12 EP claimed
US-20110118257-A1 NOVEL KINASE MODULATORS RHIZEN PHARMACEUTICALS SA (CH) 2011-05-19 US claimed
WO-2011055215-A2 NOVEL KINASE MODULATORS INCOZEN THERAPEUTICS PVT. LTD. (IN) 2011-05-12 WO claimed
US-20240360095-A1 NOVEL KINASE MODULATORS RHIZEN PHARMACEUTICALS AG (CH) 2024-10-31 US disclosed
US-20240139198-A1 METHOD AND COMBINATION FOR TREATING TUMORS CURON BIOPHARMACEUTICAL (SHANGHAI) CO., LIMITED (CN) 2024-05-02 US disclosed
US-11858907-B2 Kinase modulators RHIZEN PHARMACEUTICALS AG (CH) 2024-01-02 US disclosed
US-11858907-B2 Kinase modulators RHIZEN PHARMACEUTICALS AG (CH) 2024-01-02 US disclosed
US-11858907-B2 Kinase modulators RHIZEN PHARMACEUTICALS AG (CH) 2024-01-02 US disclosed
EP-4292596-A1 METHOD AND COMBINATION FOR TREATING TUMORS Curon Biopharmaceutical (Shanghai) Co., Limited (CN) 2023-12-20 EP disclosed
US-20120059001-A1 NOVEL KINASE MODULATORS INCOZEN THERAPEUTICS PVT. LTD. (IN) 2012-03-08 US disclosed
US-20110118257-A1 NOVEL KINASE MODULATORS RHIZEN PHARMACEUTICALS SA (CH) 2011-05-19 US disclosed
US-20110118257-A1 NOVEL KINASE MODULATORS RHIZEN PHARMACEUTICALS SA (CH) 2011-05-19 US disclosed
US-20110118257-A1 NOVEL KINASE MODULATORS RHIZEN PHARMACEUTICALS SA (CH) 2011-05-19 US disclosed
WO-2011055215-A2 NOVEL KINASE MODULATORS INCOZEN THERAPEUTICS PVT. LTD. (IN) 2011-05-12 WO disclosed
WO-2011055215-A2 NOVEL KINASE MODULATORS INCOZEN THERAPEUTICS PVT. LTD. (IN) 2011-05-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240360095-A1 NOVEL KINASE MODULATORS PRKCA, PRKCH, PRKCB NPC1 1419/4885RAB9A 1297/4885ATM 355/4885
US-20110118257-A1 NOVEL KINASE MODULATORS PRKCA, PRKCH, PRKCB NPC1 1419/4885RAB9A 1297/4885ATM 355/4885
US-20200239427-A1 NOVEL KINASE MODULATORS PRKCA, PRKCH, PRKCB NPC1 1419/4885RAB9A 1297/4885ATM 355/4885
US-11858907-B2 Kinase modulators RPS6KA1, RPS6KA2, PRKAR2A NPC1 2061/4885RAB9A 1518/4885ATM 392/4885
US-20240139198-A1 METHOD AND COMBINATION FOR TREATING TUMORS PDCD1, PDCD1LG2, CD274 NPC1 3045/4885RAB9A 2658/4885ATM 119/4885
US-20120059001-A1 NOVEL KINASE MODULATORS PRKCA, PRKCH, PRKCB NPC1 1419/4885RAB9A 1297/4885ATM 355/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.