SCHEMBL825518

SCHEMBL825518

CCOC(C[SiH2]CCCNc1ccccc1)OCC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.47
ALDH1A1 P00352 1/20 0.47
KCNH3 Q9ULD8 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
EPHX1 P07099 1/20 0.34
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
NCOR2 Q9Y618 1/20 0.33
NPC1 O15118 1/20 0.33
USP2 O75604 1/20 0.33
TP53 P04637 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HRH3 Q9Y5N1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL825907 0.83 MAPT (0.36) MAPTALDH1A1L3MBTL1CYP1A2CYP3A4
SCHEMBL1021962 0.80 MAPT (0.48) MAPTALDH1A1KCNH3L3MBTL1CYP1A2
SCHEMBL19838187 0.75 CYP2C19 (0.32) ALDH1A1CYP1A2CYP2C19
SCHEMBL1603893 0.74 ALDH1A1 (0.53) MAPTALDH1A1KCNH3L3MBTL1CYP1A2
SCHEMBL28000120 0.74 MAPT (0.39) MAPTALDH1A1KCNH3CYP1A2CYP3A4
SCHEMBL16197517 0.73 EPHX1 (0.33) EPHX1
SCHEMBL935506 0.73 MAPT (0.49) MAPTALDH1A1L3MBTL1EPHX1SMN1; SMN2
SCHEMBL704452 0.72 THRB (0.36)
SCHEMBL702536 0.72 THRB (0.36)
SCHEMBL29162935 0.71 MAPT (0.64) MAPTALDH1A1KCNH3L3MBTL1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3157970-B1 SILYLATED POLYURETHANES HUNTSMAN INT LLC (US) 2019-02-06 EP claimed
EP-3157970-A1 SILYLATED POLYURETHANES Huntsman International LLC (US) 2017-04-26 EP claimed
WO-2015193146-A1 SILYLATED POLYURETHANES HUNTSMAN INTERNATIONAL LLC (US) 2015-12-23 WO claimed
EP-3157970-A1 SILYLATED POLYURETHANES Huntsman International LLC (US) 2017-04-26 EP disclosed
WO-2015193146-A1 SILYLATED POLYURETHANES HUNTSMAN INTERNATIONAL LLC (US) 2015-12-23 WO disclosed
EP-2582737-A1 ALKOXYSILANE FUNCTIONALIZED ISOCYANATE BASED MATERIALS Huntsman International LLC (US) 2013-04-24 EP disclosed
WO-2011161011-A1 ALKOXYSILANE FUNCTIONALIZED ISOCYANATE BASED MATERIALS HUNTSMAN INTERNATIONAL LLC (US) 2011-12-29 WO disclosed