SCHEMBL8259077

SCHEMBL8259077

Cc1nc(-c2ccccc2)c(NC(=O)NS(=O)(=O)c2cnc3ccccn23)s1

nearest known ligand 0.71

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 16/20 0.71
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
PKM P14618 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
POLB P06746 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16586722 0.77 NTRK1 (1.00) NTRK1ALDH1A1KDM4EPKMHPGD
SCHEMBL16595137 0.75 NTRK1 (1.00) NTRK1ALDH1A1KDM4EHSD17B10POLB
SCHEMBL5815917 0.74 NTRK1 (0.65) NTRK1ALDH1A1KDM4EGAAMAPT
SCHEMBL5813841 0.73 NTRK1 (0.60) NTRK1ALDH1A1KDM4EPOLBGAA
SCHEMBL5814366 0.73 NTRK1 (0.57) NTRK1ALDH1A1KDM4EPOLBGAA
SCHEMBL5819741 0.73 NTRK1 (0.57) NTRK1ALDH1A1KDM4EPOLBGAA
SCHEMBL8827534 0.73 GAA (0.54) ALDH1A1KDM4EPKMHPGDHSD17B10
SCHEMBL5804272 0.73 NTRK1 (0.62) NTRK1ALDH1A1KDM4EPOLBGAA
SCHEMBL8252821 0.71 NTRK1 (0.60) NTRK1ALDH1A1GAA
SCHEMBL5814359 0.71 NTRK1 (0.85) NTRK1ALDH1A1KDM4EHSD17B10POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006085815-A1 THIAZOLE DERIVATIVES, THEIR PROCESS FOR THEIR PREPARATION AND THEIR USE IN THERAPY ASTRAZENECA AB (SE) 2006-08-17 WO disclosed