SCHEMBL8259404

SCHEMBL8259404

C=C(Cl)C(=C)C(=O)Nc1ccc(C[C@H](NC(=O)C2C3CCC(CC3)N2C(=O)OCc2ccccc2)C(=O)OC)cc1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.44
TSHR P16473 3/20 0.44
ALDH1A1 P00352 2/20 0.44
ITGB1 P05556 12/20 0.42
ITGA4 P13612 12/20 0.42
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
GAA P10253 1/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8293264 0.85 MDM4 (0.49) CYP3A4TSHRALDH1A1ITGB1ITGA4
SCHEMBL5805018 0.84 CYP3A4 (0.47) CYP3A4TSHRALDH1A1ITGB1ITGA4
SCHEMBL8254376 0.84 CYP3A4 (0.47) CYP3A4TSHRALDH1A1ITGB1ITGA4
SCHEMBL8258817 0.83 ITGB1 (0.52) ITGB1ITGA4
SCHEMBL5806399 0.83 ITGB1 (0.52) ITGB1ITGA4
SCHEMBL5910985 0.81 CYP3A4 (0.44) CYP3A4TSHRALDH1A1ITGB1ITGA4
SCHEMBL8259306 0.81 CYP3A4 (0.44) CYP3A4TSHRALDH1A1ITGB1ITGA4
SCHEMBL8293260 0.77 YAP1 (0.46) CYP3A4TSHRALDH1A1MEN1KMT2A
SCHEMBL24945845 0.70 ITGA4 (0.69) ITGB1ITGA4
SCHEMBL8259308 0.68 AGTR2 (0.56) ALDH1A1MEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006096807-A1 AZA-BRIDGED-BICYCLIC AMINO ACID DERIVATIVES AS ALPHA 4 INTEGRIN ANTAGONISTS JANSSEN PHARMACEUTICA N.V. (BE) 2006-09-14 WO disclosed