SCHEMBL8263299

SCHEMBL8263299

CC(C)(C)OC(=O)N1CCC(NCCCOc2ccc3c(c2)[nH]c2ccccc23)CC1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.48
VCP P55072 2/20 0.46
GPR119 Q8TDV5 9/20 0.45
ALDH1A1 P00352 1/20 0.44
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
KIT P10721 1/20 0.43
FLT3 P36888 1/20 0.43
PARP1 P09874 1/20 0.43
PRMT5 O14744 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14023045 0.85 ADRB3 (0.49) VCPALDH1A1
SCHEMBL8262374 0.84 ADRB2 (0.48) MCL1VCPPARP1
SCHEMBL24302272 0.78 ALDH1A1 (0.51) GPR119ALDH1A1
SCHEMBL28943536 0.75 PARP1 (0.52) GPR119ALDH1A1PARP1
SCHEMBL23635039 0.74 GPR119 (0.43) GPR119ALDH1A1PDE3BPDE3A
SCHEMBL4213070 0.73 DRD4 (0.57) GPR119ALDH1A1
SCHEMBL8267242 0.73 KDM4E (0.50) GPR119ALDH1A1
SCHEMBL8263806 0.71 ADRB3 (0.65)
SCHEMBL4899642 0.71 ADRB3 (0.65)
SCHEMBL4902486 0.71 ADRB3 (0.65)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006060122-A9 CARDIOTONIC COMPOUNDS WITH INHIBITORY ACTIVITY AGAINST BETA-ADRENERGIC RECEPTORS AND PHOSPHODIESTERASE ARTESIAN THERAPEUTICS INC (US) 2006-08-17 WO disclosed
WO-2006060122-A2 CARDIOTONIC COMPOUNDS WITH INHIBITORY ACTIVITY AGAINST BETA-ADRENERGIC RECEPTORS AND PHOSPHODIESTERASE ARTESIAN THERAPEUTICS, INC. (US) 2006-06-08 WO disclosed