SCHEMBL8265377

SCHEMBL8265377

CSc1cc(CF)cc(C(F)(F)F)c1C(=O)NC(c1ccccc1)C(C)(C)N1CCCC1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 9/20 0.36
SLC6A9 P48067 5/20 0.34
TACR3 P29371 2/20 0.33
NR1I2 O75469 1/20 0.33
TACR1 P25103 1/20 0.33
TACR2 P21452 1/20 0.33
KCNH2 Q12809 1/20 0.33
CACNA1C Q13936 1/20 0.33
SCN5A Q14524 1/20 0.33
CCR2 P41597 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
SLC6A5 Q9Y345 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3236142 0.88 SLC6A9 (0.41) TRPV4SLC6A9TACR3TACR1CYP2D6
SCHEMBL3240772 0.80 SLC6A9 (0.45) TRPV4SLC6A9
SCHEMBL3244977 0.78 TACR1 (0.39) TRPV4SLC6A9TACR3TACR1
SCHEMBL3238790 0.77 LMNA (0.35) SLC6A9CYP2D6
SCHEMBL5353056 0.76 SLC6A9 (0.42) SLC6A9CYP2D6CYP2C19SLC6A5
SCHEMBL3238426 0.76 SLC6A9 (0.42) SLC6A9CYP2C19SLC6A5
SCHEMBL3238049 0.76 ITGA4 (0.49) SLC6A9
SCHEMBL13303995 0.76 MTTP (0.40) TRPV4TACR3TACR1CCR2
SCHEMBL3832646 0.75 SLC6A9 (0.52) SLC6A9TACR1CYP2D6CYP2C19SLC6A5
SCHEMBL3008740 0.75 SLC6A9 (0.52) SLC6A9TACR1CYP2D6CYP2C19SLC6A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006067423-A1 GLYCINE TRANSPORT INHIBITORS GLAXO GROUP LIMITED (GB) 2006-06-29 WO disclosed