SCHEMBL5353056

SCHEMBL5353056

COc1cc(F)cc(SC)c1C(=O)NC(c1ccccc1)C(C)(C)N1CCCC1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 14/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
SLC6A5 Q9Y345 1/20 0.42
ROCK2 O75116 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3237806 0.89 ROCK2 (0.43) SLC6A9ROCK2
SCHEMBL12132690 0.87 SLC6A9 (0.40) SLC6A9CYP2D6CYP2C19SLC6A5
SCHEMBL5363493 0.84 ROCK2 (0.38) SLC6A9CYP2D6CYP2C19SLC6A5ROCK2
SCHEMBL3239591 0.81 KMT2A (0.47) SLC6A9CYP2D6
SCHEMBL3238200 0.80 CCR5 (0.39) SLC6A9CYP2C19SLC6A5
SCHEMBL26840793 0.80 RXFP1 (0.38) SLC6A9
SCHEMBL3236158 0.79 SLC6A9 (0.41) SLC6A9
SCHEMBL1350280 0.79 SLC6A9 (0.45) SLC6A9CYP2D6CYP2C19SLC6A5ROCK2
SCHEMBL3236142 0.79 SLC6A9 (0.41) SLC6A9CYP2D6CYP2C19SLC6A5
SCHEMBL3008740 0.79 SLC6A9 (0.52) SLC6A9CYP2D6CYP2C19SLC6A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007147834-A1 GLYCINE TRANSPORTER INHIBITING COMPOUNDS AND USES IN MEDICINE GLAXO GROUP LIMITED (GB) 2007-12-27 WO claimed
WO-2007147834-A1 GLYCINE TRANSPORTER INHIBITING COMPOUNDS AND USES IN MEDICINE GLAXO GROUP LIMITED (GB) 2007-12-27 WO disclosed
WO-2007147834-A1 GLYCINE TRANSPORTER INHIBITING COMPOUNDS AND USES IN MEDICINE GLAXO GROUP LIMITED (GB) 2007-12-27 WO disclosed