SCHEMBL8268115

SCHEMBL8268115

CC(C)Oc1cccc(CN2CCC3(CC2)C(NC2CCCCC2)=NC(=O)N3c2ccccc2-c2ccc(CN)cc2)c1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MLNR O43193 1/20 0.37
FAAH O00519 1/20 0.36
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
ADRA1D P25100 1/20 0.35
HTR1B P28222 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35
DRD3 P35462 1/20 0.35
SSTR5 P35346 1/20 0.35
CCR8 P51685 1/20 0.35
HRH2 P25021 1/20 0.35
CCKBR P32239 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL593096 0.93 MLNR (0.36) MLNRFAAHHTR1ADRD2ADRA1D
SCHEMBL593208 0.92 CCR5 (0.39) HTR1ADRD2ADRA1DHTR1BADRA1A
SCHEMBL593105 0.91 FAAH (0.35) MLNRFAAHHTR1ADRD2ADRA1D
SCHEMBL593094 0.91 CXCR3 (0.38) FAAHDRD2
SCHEMBL594223 0.91 HTR1A (0.37) MLNRFAAHHTR1ADRD2ADRA1D
SCHEMBL593551 0.91 CCR5 (0.41)
SCHEMBL593104 0.90 FAAH (0.33) MLNRFAAHHTR1ADRD2ADRA1D
SCHEMBL594222 0.89 MLNR (0.35) MLNRFAAHHTR1ADRD2ADRA1D
SCHEMBL594391 0.88 OPRL1 (0.39) FAAH
SCHEMBL593097 0.88 MAP3K11 (0.38) MLNRFAAHSSTR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006044497-A2 SPIROPIPERIDINE COMPOUNDS USEFUL AS BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHERMER’S DISEASE MERCK & CO., INC. (US) 2006-04-27 WO disclosed