SCHEMBL8274181

SCHEMBL8274181

NCOBCc1ccc(C(=O)N2CC(O)C2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR2 O60603 1/20 0.39
TLR1 Q15399 1/20 0.39
VNN1 O95497 1/20 0.36
HSD11B1 P28845 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.36
PDK2 Q15119 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA7 P36544 1/20 0.35
CHRNA4 P43681 1/20 0.35
ALDH1A1 P00352 2/20 0.34
HPGD P15428 1/20 0.34
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34
GRM3 Q14832 1/20 0.34
CCNC P24863 2/20 0.34
CDK8 P49336 2/20 0.34
L3MBTL3 Q96JM7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8275305 0.87 GRM5 (0.47) HSD11B1ALDH1A1HPGDMAPTGRM3
SCHEMBL12163055 0.85 MRGPRX4 (0.49) VNN1MRGPRX4PDK2ALDH1A1NPC1
SCHEMBL8275216 0.83 HPGD (0.53) ALDH1A1HPGDNPC1MAPTRAB9A
SCHEMBL8275217 0.81 ALDH1A1 (0.48) HSD11B1ALDH1A1HPGDNPC1MAPT
SCHEMBL12162954 0.81 ALDH1A1 (0.48) HSD11B1ALDH1A1HPGDNPC1MAPT
SCHEMBL8274693 0.79 HDAC3 (0.44) TLR2TLR1VNN1PDK2CHRNB2
SCHEMBL8275193 0.77 RORC (0.34)
SCHEMBL12162956 0.76 LOXL2 (0.50) VNN1MRGPRX4PDK2HPGDNPC1
SCHEMBL17850465 0.73 ALDH1A1 (0.48) TLR2TLR1ALDH1A1HPGDMAPT
SCHEMBL8275220 0.72 MRGPRX4 (0.36) MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005116009-A1 SUBSTITUTED 2-QUINOLYL-OXAZOLES USEFUL AS PDE4 INHIBITORS SCHERING CORPORATION (US) 2005-12-08 WO disclosed