SCHEMBL8278122

SCHEMBL8278122

CCc1ccc2c(c1)[C@H](NC(C)=O)[C@@H](Br)CO2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
CASP6 P55212 1/20 0.39
HKDC1 Q2TB90 1/20 0.39
MTNR1A P48039 4/20 0.37
TP53 P04637 2/20 0.36
DRD2 P14416 4/20 0.35
DRD3 P35462 4/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
AIMP2 Q13155 1/20 0.35
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8278101 0.77 HCRTR2 (0.44) HCRTR2KDM4EALDH1A1TP53DRD2
SCHEMBL7757152 0.72 MTNR1A (0.50) HCRTR2MEN1KMT2AMTNR1ATP53
SCHEMBL13038051 0.69 HCRTR2 (0.48) HCRTR2KDM4EALDH1A1TP53DRD2
SCHEMBL22923302 0.69 HCRTR2 (0.48) HCRTR2KDM4EALDH1A1TP53DRD2
SCHEMBL8278342 0.66 HCRTR2 (0.44) HCRTR2ALDH1A1MEN1KMT2ATP53
SCHEMBL5713612 0.66 HCRTR2 (0.44) HCRTR2ALDH1A1MEN1KMT2ATP53
SCHEMBL9581223 0.65 HCRTR2 (0.43) HCRTR2KDM4EALDH1A1TP53DRD2
SCHEMBL11864992 0.64 HCRTR2 (0.43) HCRTR2MEN1KMT2ATP53CYP1A2
SCHEMBL25146821 0.64 PPARG (0.56)
SCHEMBL8126531 0.64 HCRTR2 (0.42) HCRTR2KDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100145056-A1 ACETYL 2-HYDROXY-1,3-DIAMINOALKANES JOHN VARGHESE 2010-06-10 US disclosed
US-7645780-B2 Acetyl 2-hydroxy-1, 3-diaminoalkanes ELAN PHARMACEUTICALS, INC. (US) 2010-01-12 US disclosed
US-7544717-B2 2-amino- and 2-thio- substituted 1,3-diaminopropanes ELAN PHARMACEUTICALS, INC. (US) 2009-06-09 US disclosed
US-20070293483-A1 Acetyl 2-hydroxy-1, 3-diaminoalkanes ELAN PHARMACEUTICALS, INC. 2007-12-20 US disclosed
US-7244725-B2 Acetyl 2-hydroxy-1, 3-diaminoalkanes ELAN PHARMACEUTICALS, INC. (US) 2007-07-17 US disclosed
WO-2005087714-A2 METHODS OF TREATMENT OF AMYLOIDOSIS USING BI-CYCLIC ASPARTYL PROTEASE INHIBITORS ELAN PHARMACEUTICALS, INC. (US) 2005-09-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100145056-A1 ACETYL 2-HYDROXY-1,3-DIAMINOALKANES BACE1, BACE2, APP HCRTR2 215/4885KDM4E 3339/4885ALDH1A1 638/4885
US-20070293483-A1 Acetyl 2-hydroxy-1, 3-diaminoalkanes BACE1, BACE2, APP HCRTR2 215/4885KDM4E 3339/4885ALDH1A1 638/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.