SCHEMBL8278796

SCHEMBL8278796

N#Cc1c(Cl)ccc([N+](=O)[O-])c1NCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.47
VCAM1 P19320 2/20 0.46
MAPT P10636 5/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
NPC1 O15118 1/20 0.44
TLR9 Q9NR96 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
USP2 O75604 1/20 0.43
HTT P42858 1/20 0.43
RECQL P46063 1/20 0.43
PTPRF P10586 1/20 0.43
PTPN2 P17706 1/20 0.43
PTPN1 P18031 1/20 0.43
PTPN11 Q06124 1/20 0.43
HTR6 P50406 2/20 0.42
POLB P06746 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP1A2 P05177 3/20 0.41
CYP3A4 P08684 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3149356 0.87 RAB9A (0.43) RAB9AVCAM1MAPTL3MBTL1NPC1
SCHEMBL3153199 0.81 RAB9A (0.51) RAB9AVCAM1MAPTMEN1KMT2A
SCHEMBL7779674 0.81 RAB9A (0.51) RAB9AVCAM1MAPTNPC1MEN1
SCHEMBL3149349 0.79 RAB9A (0.74) RAB9AVCAM1MAPTL3MBTL1MEN1
SCHEMBL894368 0.76 VCAM1 (0.47) RAB9AVCAM1MAPTPOLBLMNA
SCHEMBL25352613 0.73 VCAM1 (0.44) RAB9AVCAM1MAPTNPC1SMN1; SMN2
SCHEMBL8313813 0.72 VCAM1 (0.56) RAB9AVCAM1MAPTHPGDALDH1A1
SCHEMBL29411983 0.71 HTR6 (0.58) MAPTL3MBTL1MEN1KMT2AUSP2
SCHEMBL894816 0.71 TDP1 (0.60) RAB9AVCAM1MAPTPOLBCYP2C9
SCHEMBL272708 0.71 TDP1 (0.60) RAB9AVCAM1MAPTHPGDEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7687638-B2 Dipeptidyl peptidase inhibitors TAKEDA SAN DIEGO, INC. (US) 2010-03-30 US disclosed
US-7687638-B2 Dipeptidyl peptidase inhibitors TAKEDA SAN DIEGO, INC. (US) 2010-03-30 US disclosed
WO-2005118555-A1 DIPEPTIDYL PEPTIDASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-12-15 WO disclosed