SCHEMBL828014

SCHEMBL828014

CCN(C(=O)O)c1ccc2cc(-c3ccccc3N3CCOCC3)[nH]c(=O)c2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APAF1 O14727 1/20 0.40
CDC25B P30305 1/20 0.40
CASP3 P42574 1/20 0.40
SENP8 Q96LD8 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
ALDH1A1 P00352 3/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
MDM2 Q00987 1/20 0.40
AKT1 P31749 11/20 0.40
BRD4 O60885 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
GAA P10253 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
KDM4C Q9H3R0 1/20 0.37
PIK3CD O00329 4/20 0.37
PIK3CA P42336 4/20 0.37
PIK3CB P42338 4/20 0.37
PIK3CG P48736 4/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL828336 0.79 TNKS (0.48) APAF1CASP3SENP8SENP7ALDH1A1
SCHEMBL826935 0.78 FFAR1 (0.44) APAF1CASP3SENP8SENP7ALDH1A1
SCHEMBL2711139 0.78 APAF1 (0.46) APAF1CDC25BCASP3SENP8SENP7
SCHEMBL824947 0.78 TDO2 (0.51) APAF1CDC25BCASP3SENP8SENP7
SCHEMBL824701 0.77 APAF1 (0.49) APAF1CDC25BCASP3SENP8SENP7
SCHEMBL824716 0.77 APAF1 (0.49) APAF1CDC25BCASP3SENP8SENP7
SCHEMBL824737 0.76 NR1I3 (0.49) APAF1CDC25BCASP3SENP8SENP7
SCHEMBL827412 0.76 FFAR1 (0.46) APAF1CASP3SENP8SENP7ALDH1A1
SCHEMBL824950 0.75 TDO2 (0.48) APAF1CDC25BCASP3SENP8SENP7
SCHEMBL824945 0.74 TDO2 (0.47) APAF1CDC25BCASP3SENP8SENP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143274-B2 1-(2H)-isoquinolone derivative CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2012-03-27 US disclosed