SCHEMBL8288343

SCHEMBL8288343

C=C1OB(c2ccc(CCNS(=O)(=O)c3cccc(F)c3)cc2)OC1=C

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
PRMT1 Q99873 1/20 0.45
TAAR1 Q96RJ0 1/20 0.45
AKR1C3 P42330 4/20 0.44
KMT2A Q03164 2/20 0.42
MAPK1 P28482 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
SOST Q9BQB4 1/20 0.41
GBA1 P04062 1/20 0.40
POLB P06746 1/20 0.40
SGMS1 Q86VZ5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8287312 0.86 AKR1C3 (0.51) ALDH1A1PRMT1AKR1C3KMT2AMAPK1
SCHEMBL8288311 0.86 TAAR1 (0.59) ALDH1A1TAAR1KMT2ATDP1CA1
SCHEMBL8289277 0.86 ALDH1A1 (0.57) ALDH1A1PRMT1TAAR1AKR1C3KMT2A
SCHEMBL13612187 0.84 ALDH1A1 (0.42) ALDH1A1PRMT1TAAR1AKR1C3KMT2A
SCHEMBL8289264 0.84 LSS (0.43) ALDH1A1PRMT1AKR1C3KMT2AMAPK1
SCHEMBL13604124 0.83 CA1 (0.47) ALDH1A1PRMT1TAAR1AKR1C3KMT2A
SCHEMBL8288351 0.79 TP53 (0.42) ALDH1A1TAAR1KMT2ACA1CA2
SCHEMBL8287311 0.79 ALDH1A1 (0.68) ALDH1A1AKR1C3KMT2ACA1CA2
SCHEMBL13611732 0.79 MEN1 (0.60) ALDH1A1PRMT1AKR1C3KMT2ACA1
SCHEMBL8288312 0.76 LSS (0.56) ALDH1A1TAAR1KMT2ACA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1670757-B1 PYRROLE AND PYRAZOLE DERIVATIVES AS POTENTIATORS OF GLUTAMATE RECEPTORS LILLY CO ELI (US) 2009-05-06 EP disclosed
WO-2005040110-A1 PYRROLE AND PYRAZOLE DERIVATIVES AS POTENTIATORS OF GLUTAMATE RECEPTORS ELI LILLY AND COMPANY (US) 2005-05-06 WO disclosed