SCHEMBL8288351

SCHEMBL8288351

C=C1OB(c2ccc(CCNS(=O)(=O)c3ccccc3F)cc2)OC1=C

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.42
TAAR1 Q96RJ0 1/20 0.41
ALDH1A1 P00352 3/20 0.40
NSD2 O96028 2/20 0.40
TSHR P16473 1/20 0.40
GBA1 P04062 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GRIA4 P48058 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8288313 0.86 CA1 (0.42) ALDH1A1NSD2SMN1; SMN2KMT2ACA1
SCHEMBL13611592 0.84 TP53 (0.40) TP53TAAR1ALDH1A1NSD2TSHR
SCHEMBL8288305 0.83 SMN1; SMN2 (0.39) ALDH1A1NSD2SMN1; SMN2KMT2ACA1
SCHEMBL8289277 0.83 ALDH1A1 (0.57) TAAR1ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL13604122 0.82 LPL (0.47) TP53TAAR1ALDH1A1TSHRGRIA4
SCHEMBL8288311 0.81 TAAR1 (0.59) TAAR1ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL8288343 0.79 ALDH1A1 (0.45) TAAR1ALDH1A1GBA1KMT2ACA1
SCHEMBL8289308 0.76 PKM (0.59) TP53ALDH1A1TSHRHTT
SCHEMBL8287311 0.76 ALDH1A1 (0.68) TP53ALDH1A1TSHRSMN1; SMN2MEN1
SCHEMBL13611732 0.76 MEN1 (0.60) TP53ALDH1A1SMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1670757-B1 PYRROLE AND PYRAZOLE DERIVATIVES AS POTENTIATORS OF GLUTAMATE RECEPTORS LILLY CO ELI (US) 2009-05-06 EP disclosed
WO-2005040110-A1 PYRROLE AND PYRAZOLE DERIVATIVES AS POTENTIATORS OF GLUTAMATE RECEPTORS ELI LILLY AND COMPANY (US) 2005-05-06 WO disclosed