SCHEMBL8289264

SCHEMBL8289264

C=C1OB(c2ccc(CCNS(=O)(=O)c3cccc(C#N)c3)cc2)OC1=C

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LSS P48449 2/20 0.43
ALDH1A1 P00352 2/20 0.43
PRMT1 Q99873 1/20 0.43
AKR1C3 P42330 4/20 0.41
MAPK1 P28482 1/20 0.40
KMT2A Q03164 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
HDAC2 Q92769 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CYP19A1 P11511 1/20 0.39
F10 P00742 1/20 0.38
PRSS1 P07477 1/20 0.38
PRSS2 P07478 1/20 0.38
PRSS3 P35030 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8288312 0.87 LSS (0.56) LSSALDH1A1KMT2ACA1CA2
SCHEMBL13611590 0.85 ALDH1A1 (0.40) LSSALDH1A1PRMT1AKR1C3MAPK1
SCHEMBL8288343 0.84 ALDH1A1 (0.45) ALDH1A1PRMT1AKR1C3MAPK1KMT2A
SCHEMBL8287312 0.84 AKR1C3 (0.51) ALDH1A1PRMT1AKR1C3MAPK1KMT2A
SCHEMBL8289277 0.83 ALDH1A1 (0.57) ALDH1A1PRMT1AKR1C3KMT2ATDP1
Water SCHEMBL28775032 0.79 ALDH1A1 (0.50) LSSALDH1A1PRMT1AKR1C3MAPK1
SCHEMBL3861652 0.79 LSS (0.50) LSSALDH1A1PRMT1AKR1C3MAPK1
SCHEMBL8288305 0.78 SMN1; SMN2 (0.39) LSSALDH1A1KMT2ACA1CA2
SCHEMBL3861470 0.78 LSS (0.51) LSSALDH1A1PRMT1AKR1C3MAPK1
SCHEMBL13611732 0.76 MEN1 (0.60) LSSALDH1A1PRMT1AKR1C3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1670757-B1 PYRROLE AND PYRAZOLE DERIVATIVES AS POTENTIATORS OF GLUTAMATE RECEPTORS LILLY CO ELI (US) 2009-05-06 EP disclosed
WO-2005040110-A1 PYRROLE AND PYRAZOLE DERIVATIVES AS POTENTIATORS OF GLUTAMATE RECEPTORS ELI LILLY AND COMPANY (US) 2005-05-06 WO disclosed