SCHEMBL8288598

SCHEMBL8288598

CC1CCN(CCC(=O)Nc2sc3c(c2N)CCCCC3)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
TSHR P16473 2/20 0.54
KDM4E B2RXH2 1/20 0.54
ALOX15 P16050 1/20 0.54
HSD17B10 Q99714 1/20 0.54
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
RORC P51449 1/20 0.49
MAPT P10636 1/20 0.49
POLB P06746 2/20 0.49
HTT P42858 1/20 0.49
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
GAA P10253 2/20 0.46
TP53 P04637 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
HPGD P15428 2/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8289734 0.85 ALDH1A1 (0.76) ALDH1A1TSHRKDM4EALOX15HSD17B10
SCHEMBL8288576 0.77 ALDH1A1 (0.71) ALDH1A1TSHRKDM4EALOX15HSD17B10
SCHEMBL8289733 0.77 ALDH1A1 (0.71) ALDH1A1TSHRKDM4EALOX15HSD17B10
SCHEMBL5455543 0.74 ALDH1A1 (0.78) ALDH1A1TSHRKDM4EALOX15HSD17B10
SCHEMBL8290347 0.71 ALDH1A1 (0.69) ALDH1A1TSHRKDM4EALOX15HSD17B10
Oxalic Acid SCHEMBL34468543 0.68 ALDH1A1 (0.70) ALDH1A1TSHRKDM4EALOX15HSD17B10
SCHEMBL8288703 0.68 LMNA (0.47) ALDH1A1TSHRKDM4EMEN1KMT2A
SCHEMBL15369925 0.68 POLB (1.00) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL34468524 0.68 KMT2A (0.83) ALDH1A1TSHRKDM4EALOX15HSD17B10
SCHEMBL8288718 0.67 MEN1 (0.96) ALDH1A1TSHRKDM4EALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed