SCHEMBL8288763

SCHEMBL8288763

CCCS(=O)(=O)Nc1scc(-c2ccc(OC)c(OC)c2)c1C(=O)OCC

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 9/20 0.64
ALDH1A1 P00352 5/20 0.57
HTT P42858 4/20 0.57
CRHBP P24387 1/20 0.57
CRHR2 Q13324 1/20 0.57
PRKCZ Q05513 5/20 0.52
HPGD P15428 3/20 0.50
MAPK1 P28482 1/20 0.50
HSD17B10 Q99714 1/20 0.50
NPC1 O15118 1/20 0.49
LMNA P02545 3/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
NPSR1 Q6W5P4 2/20 0.48
PTPN1 P18031 1/20 0.48
KDM4E B2RXH2 2/20 0.46
MEN1 O00255 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13837645 0.82 MAPT (0.76) MAPTALDH1A1HTTCRHBPCRHR2
SCHEMBL8290370 0.81 MAPT (0.68) MAPTALDH1A1HTTCRHBPCRHR2
SCHEMBL5804278 0.81 MAPT (0.73) MAPTALDH1A1HTTCRHBPCRHR2
SCHEMBL5804285 0.80 MAPT (0.72) MAPTALDH1A1HTTCRHBPCRHR2
SCHEMBL8288714 0.77 PRKCZ (0.81) MAPTALDH1A1PRKCZHPGDMAPK1
SCHEMBL7970089 0.70 HTT (0.53) MAPTALDH1A1HTTCRHBPCRHR2
SCHEMBL13837727 0.68 PRKCZ (1.00) MAPTALDH1A1PRKCZHPGDMAPK1
SCHEMBL1895353 0.68 MEN1 (0.78) MAPTALDH1A1CRHBPCRHR2HPGD
SCHEMBL10459766 0.68 HTT (0.56) MAPTALDH1A1HTTPRKCZHPGD
SCHEMBL7980488 0.68 HTT (0.60) MAPTALDH1A1HTTPRKCZHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed