SCHEMBL8290603

SCHEMBL8290603

CCCC1CCc2c(sc(NC(=O)c3ccncc3)c2C(N)=O)C1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.72
KDM4E B2RXH2 6/20 0.72
RAB9A P51151 4/20 0.72
HPGD P15428 4/20 0.72
NPC1 O15118 3/20 0.72
NPSR1 Q6W5P4 1/20 0.72
MAPT P10636 5/20 0.69
KMT2A Q03164 3/20 0.69
PDE4B Q07343 3/20 0.69
PDE4D Q08499 3/20 0.69
SMN1; SMN2 Q16637 3/20 0.62
FLT3 P36888 2/20 0.62
POLB P06746 1/20 0.61
REV1 Q9UBZ9 1/20 0.58
MEN1 O00255 2/20 0.57
TP53 P04637 1/20 0.57
HTT P42858 1/20 0.57
USP2 O75604 1/20 0.56
XBP1 P17861 1/20 0.56
HSD17B10 Q99714 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8289821 0.85 MAPT (0.76) ALDH1A1KDM4ERAB9ANPC1MAPT
SCHEMBL4145641 0.83 MAPT (0.82) ALDH1A1KDM4ERAB9AHPGDNPC1
SCHEMBL21346802 0.82 MAPT (1.00) ALDH1A1KDM4ERAB9AHPGDNPC1
SCHEMBL21347427 0.82 MAPT (1.00) ALDH1A1KDM4ERAB9AHPGDNPC1
SCHEMBL21347434 0.82 ALDH1A1 (0.62) ALDH1A1KDM4ERAB9AHPGDNPC1
SCHEMBL5454136 0.80 REV1 (0.81) ALDH1A1KDM4ERAB9AHPGDNPC1
SCHEMBL21346848 0.79 PDE4B (0.68) ALDH1A1KDM4ERAB9AHPGDNPC1
SCHEMBL1066142 0.78 FLT3 (0.68) ALDH1A1KDM4ERAB9AHPGDNPC1
SCHEMBL5457818 0.78 FLT3 (1.00) ALDH1A1RAB9ANPC1MAPTKMT2A
SCHEMBL16596087 0.76 REV1 (0.62) ALDH1A1KDM4ERAB9AHPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed