SCHEMBL8290684

SCHEMBL8290684

CCOC(=O)c1c(N)sc(C(=O)Nc2cccc(OC)c2)c1C

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CISD2 Q8N5K1 9/20 0.83
ALDH1A1 P00352 5/20 0.77
RAB9A P51151 4/20 0.77
NPC1 O15118 4/20 0.77
MAPT P10636 4/20 0.77
NFKB1 P19838 3/20 0.77
NFKB2 Q00653 3/20 0.77
RELA Q04206 3/20 0.77
SETD7 Q8WTS6 4/20 0.74
SMN1; SMN2 Q16637 2/20 0.65
MEN1 O00255 2/20 0.65
KMT2A Q03164 2/20 0.65
TP53 P04637 1/20 0.65
POLB P06746 1/20 0.65
PKM P14618 1/20 0.65
HPGD P15428 1/20 0.65
NPSR1 Q6W5P4 1/20 0.65
GUSB P08236 1/20 0.57
GAA P10253 1/20 0.56
HTT P42858 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25106688 0.89 RAB9A (0.77) CISD2ALDH1A1RAB9ANPC1MAPT
SCHEMBL9400304 0.87 RAB9A (1.00) CISD2ALDH1A1RAB9ANPC1MAPT
SCHEMBL23657451 0.85 RAB9A (0.71) CISD2ALDH1A1RAB9ANPC1MAPT
SCHEMBL13236165 0.83 ALDH1A1 (0.76) CISD2ALDH1A1RAB9ANPC1MAPT
SCHEMBL25106697 0.83 CISD2 (0.80) CISD2ALDH1A1RAB9ANPC1MAPT
SCHEMBL25106677 0.81 CISD2 (1.00) CISD2ALDH1A1RAB9ANPC1MAPT
SCHEMBL25106678 0.81 CISD2 (1.00) CISD2ALDH1A1RAB9ANPC1MAPT
SCHEMBL20838890 0.81 RAB9A (0.69) CISD2ALDH1A1RAB9ANPC1MAPT
SCHEMBL8289765 0.81 ALDH1A1 (0.83) CISD2ALDH1A1RAB9ANPC1MAPT
SCHEMBL25106684 0.76 CISD2 (1.00) CISD2ALDH1A1RAB9ANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed