SCHEMBL8296371

SCHEMBL8296371

[O-][NH+]1CCCC(CCN2CCC(Cc3ccccc3)CC2)(c2ccc(Cl)c(Cl)c2)C1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 5/20 0.43
SLC6A4 P31645 5/20 0.43
TACR1 P25103 5/20 0.43
CCR3 P51677 2/20 0.42
SLC6A3 Q01959 2/20 0.42
PRMT3 O60678 1/20 0.41
CARM1 Q86X55 1/20 0.41
PRMT6 Q96LA8 1/20 0.41
PRMT1 Q99873 1/20 0.41
PRMT8 Q9NR22 1/20 0.41
CCR5 P51681 1/20 0.41
NPFFR1 Q9GZQ6 1/20 0.41
NPFFR2 Q9Y5X5 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8300496 0.82 SLC6A2 (0.54) SLC6A2SLC6A4TACR1CCR3SLC6A3
Hydrochloric Acid SCHEMBL8742517 0.81 SLC6A2 (0.53) SLC6A2SLC6A4TACR1CCR3SLC6A3
SCHEMBL8300818 0.81 CCR5 (0.43) SLC6A2SLC6A4TACR1CCR3SLC6A3
Hydrochloric Acid SCHEMBL8521991 0.80 CCR5 (0.42) SLC6A2SLC6A4TACR1CCR3SLC6A3
SCHEMBL8296084 0.78 CCR5 (0.64) TACR1CCR5
Hydrochloric Acid SCHEMBL8522900 0.78 CCR5 (0.63) TACR1CCR5
SCHEMBL8296368 0.77 TACR1 (0.50) TACR1CCR5
SCHEMBL8300814 0.76 TACR1 (0.73) TACR1CCR5
Hydrochloric Acid SCHEMBL8521990 0.75 TACR1 (0.72) TACR1CCR5
SCHEMBL8742504 0.75 CCR5 (0.51) TACR1CCR5NPFFR1NPFFR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0512901-B1 Aminated polycyclic compounds and their enantiomers, process for their preparation and pharmaceutical compositions containing them SANOFI SA (FR) 1999-06-23 EP disclosed
US-5625060-A Polycyclic amine compounds and their enantiomers, their method of preparation and pharmaceutical compositions on which they are present Sanofi, Elf (FR) 1997-04-29 US disclosed
US-5340822-A Substance P, neurokinin antagonists ELF SANOFI (FR) 1994-08-23 US disclosed
EP-0512901-A1 Aminated polycyclic compounds and their enantiomers, process for their preparation and pharmaceutical compositions containing them SANOFI (FR) 1992-11-11 EP disclosed