SCHEMBL8742504

SCHEMBL8742504

CC(C)(C)NC(=O)N1CCCC(CCN2CCC(Cc3ccccc3)CC2)(c2ccc(Cl)c(Cl)c2)C1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 2/20 0.51
TACR1 P25103 11/20 0.48
TACR2 P21452 8/20 0.48
TACR3 P29371 6/20 0.48
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
HTT P42858 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPFFR1 Q9GZQ6 1/20 0.43
NPFFR2 Q9Y5X5 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8296084 0.86 CCR5 (0.64) CCR5TACR1TACR2TACR3CYP3A4
Hydrochloric Acid SCHEMBL8522900 0.85 CCR5 (0.63) CCR5TACR1TACR2TACR3CYP3A4
SCHEMBL8300813 0.85 TACR1 (0.58) TACR1TACR2TACR3CYP3A4CYP2D6
SCHEMBL8300790 0.80 EPHX2 (0.51) TACR1TACR2TACR3CYP3A4CYP2D6
SCHEMBL8300768 0.80 TACR2 (0.69) CCR5TACR1TACR2
SCHEMBL8296058 0.76 TACR2 (0.54) CCR5TACR1TACR2TACR3CYP3A4
Hydrochloric Acid SCHEMBL8591404 0.76 TACR2 (0.53) CCR5TACR1TACR2TACR3CYP3A4
SCHEMBL8300496 0.76 SLC6A2 (0.54) CCR5TACR1CYP2D6NPFFR1NPFFR2
SCHEMBL8300814 0.75 TACR1 (0.73) CCR5TACR1TACR2TACR3
SCHEMBL8296371 0.75 SLC6A2 (0.43) CCR5TACR1ALDH1A1NPFFR1NPFFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5625060-A Polycyclic amine compounds and their enantiomers, their method of preparation and pharmaceutical compositions on which they are present Sanofi, Elf (FR) 1997-04-29 US disclosed
US-5340822-A Substance P, neurokinin antagonists ELF SANOFI (FR) 1994-08-23 US disclosed