SCHEMBL8300389

SCHEMBL8300389

CCOC(=O)C1CC2CC(=CC#N)CCC2CN1C(=O)OC

nearest known ligand 0.45

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 2/20 0.34
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
DRD3 P35462 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8300387 1.00 IDH1 (0.34) IDH1HCRTR1HCRTR2DRD3
SCHEMBL6611656 0.86 ALDH1A1 (0.30)
SCHEMBL6611658 0.86 ALDH1A1 (0.30)
SCHEMBL8291349 0.82
SCHEMBL25475425 0.82 ALDH1A1 (0.32)
SCHEMBL3302863 0.82 ALDH1A1 (0.32)
SCHEMBL7058824 0.82 ALDH1A1 (0.32)
SCHEMBL6606249 0.81 ALDH1A1 (0.34) IDH1
SCHEMBL9518658 0.79 IDH1 (0.40) IDH1
SCHEMBL9518652 0.79 IDH1 (0.40) IDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0658545-B1 Decahydro-isoquinoline derivatives LILLY CO ELI (US) 1999-09-29 EP disclosed
EP-0383504-B1 Decahydro isoquinoline derivatives, process for their preparation and use as medicines LILLY CO ELI (US) 1995-07-19 EP disclosed
EP-0658545-A1 Decahydro-isoquinoline derivatives ELI LILLY AND COMPANY (US) 1995-06-21 EP disclosed
EP-0383504-A2 Decahydro isoquinoline derivatives, process for their preparation and use as medicines ELI LILLY AND COMPANY (US) 1990-08-22 EP disclosed
US-4902695-A ISOQUINOLINE DERIVATIVES; NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY (US) 1990-02-20 US disclosed