SCHEMBL8300508

SCHEMBL8300508

CCCCC1(c2ccco2)N=C[N+](C)(c2ccc(-c3ccccc3C#N)cc2)N1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.35
PPARG P37231 2/20 0.34
USP2 O75604 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
CYP2C19 P33261 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
ESR2 Q92731 1/20 0.32
AGTR1 P30556 3/20 0.32
AGTR2 P50052 2/20 0.31
GSK3A P49840 1/20 0.31
GSK3B P49841 1/20 0.31
MMP13 P45452 1/20 0.30
AXL P30530 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8300800 0.76 ACHE (0.40) ACHEPPARGUSP2ALDH1A1CYP1A2
SCHEMBL8300512 0.75 ACHE (0.37) ACHEPPARGUSP2ALDH1A1LMNA
SCHEMBL2692039 0.64 PPARG (0.53) ACHEPPARGALDH1A1TSHRHSD17B10
SCHEMBL4253889 0.62 HSD17B10 (0.58) ACHEPPARGALDH1A1LMNACYP3A4
Decane SCHEMBL9620442 0.62 ESR2 (0.53) ACHEPPARGALDH1A1CYP1A2TSHR
Octane SCHEMBL9620215 0.62 ESR2 (0.53) ACHEPPARGALDH1A1CYP1A2TSHR
SCHEMBL6954317 0.62 HSD17B10 (0.60) ACHEPPARGALDH1A1LMNACYP3A4
SCHEMBL10718048 0.62 HSD17B10 (0.60) ACHEPPARGALDH1A1LMNACYP3A4
SCHEMBL4256521 0.62 HSD17B10 (0.60) ACHEPPARGALDH1A1LMNACYP3A4
SCHEMBL6954649 0.62 HSD17B10 (0.60) ACHEPPARGALDH1A1LMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0936221-A1 NOVEL 2,4-DIOXOPYRROLIDINE AND 2,4-DIOXOTETRAHYDROFURAN DERIVATIVES AND MEDICINES CONTAINING THE SAME AS THE ACTIVE INGREDIENT LEAD CHEMICAL COMPANY LTD. (JP) 1999-08-18 EP disclosed