SCHEMBL8300512

SCHEMBL8300512

CCCCC1(c2ccco2)N=C(C)N(c2ccc(-c3ccccc3C#N)cc2)N1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.37
USP2 O75604 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
CYP2C19 P33261 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
PPARG P37231 2/20 0.33
ESR2 Q92731 1/20 0.32
AGTR1 P30556 3/20 0.31
PTPN5 P54829 1/20 0.31
APLNR P35414 1/20 0.31
NR3C1 P04150 1/20 0.31
AGTR2 P50052 2/20 0.31
GRIA2 P42262 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8300801 0.76 ACHE (0.41) ACHEUSP2ALDH1A1CYP1A2CYP3A4
SCHEMBL8300508 0.75 ACHE (0.35) ACHEUSP2ALDH1A1LMNACYP1A2
SCHEMBL8305889 0.67 ACHE (0.37) ACHEALDH1A1PPARGESR2AGTR1
SCHEMBL8330503 0.62 ACHE (0.38) ACHEALDH1A1CYP1A2CYP3A4CYP2D6
Octane SCHEMBL9620215 0.61 ESR2 (0.53) ACHEALDH1A1CYP1A2TSHRCYP2C19
Decane SCHEMBL9620442 0.61 ESR2 (0.53) ACHEALDH1A1CYP1A2TSHRCYP2C19
SCHEMBL2692039 0.60 PPARG (0.53) ACHEALDH1A1TSHRHSD17B10PPARG
SCHEMBL4253889 0.60 HSD17B10 (0.58) ACHEALDH1A1LMNACYP3A4TSHR
SCHEMBL6959613 0.60 ESR2 (0.51) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL10589349 0.59 PPARG (0.47) ACHEPPARGESR2AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0936221-A1 NOVEL 2,4-DIOXOPYRROLIDINE AND 2,4-DIOXOTETRAHYDROFURAN DERIVATIVES AND MEDICINES CONTAINING THE SAME AS THE ACTIVE INGREDIENT LEAD CHEMICAL COMPANY LTD. (JP) 1999-08-18 EP disclosed