SCHEMBL8300800

SCHEMBL8300800

CCCCC1(CCc2ccccc2)N=C[N+](C)(c2ccc(-c3ccccc3C#N)cc2)N1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.40
PPARG P37231 2/20 0.39
FFAR1 O14842 1/20 0.36
AKR1B1 P15121 1/20 0.36
AGTR1 P30556 4/20 0.36
AGTR2 P50052 3/20 0.36
BRS3 P32247 3/20 0.34
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
CYP2C19 P33261 1/20 0.33
BLM P54132 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8304493 0.77 BRS3 (0.30) BRS3
SCHEMBL8300508 0.76 ACHE (0.35) ACHEPPARGAGTR1AGTR2ALDH1A1
SCHEMBL8300801 0.74 ACHE (0.41) ACHEPPARGFFAR1AKR1B1AGTR1
SCHEMBL2692039 0.72 PPARG (0.53) ACHEPPARGFFAR1AKR1B1AGTR1
SCHEMBL4253889 0.71 HSD17B10 (0.58) ACHEPPARGFFAR1AKR1B1AGTR1
SCHEMBL10718048 0.70 HSD17B10 (0.60) ACHEPPARGFFAR1AKR1B1AGTR1
SCHEMBL6954317 0.70 HSD17B10 (0.60) ACHEPPARGFFAR1AKR1B1AGTR1
SCHEMBL6954649 0.70 HSD17B10 (0.60) ACHEPPARGFFAR1AKR1B1AGTR1
SCHEMBL4256521 0.70 HSD17B10 (0.60) ACHEPPARGFFAR1AKR1B1AGTR1
SCHEMBL6961928 0.69 PPARG (0.59) ACHEPPARGFFAR1AKR1B1AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0936221-A1 NOVEL 2,4-DIOXOPYRROLIDINE AND 2,4-DIOXOTETRAHYDROFURAN DERIVATIVES AND MEDICINES CONTAINING THE SAME AS THE ACTIVE INGREDIENT LEAD CHEMICAL COMPANY LTD. (JP) 1999-08-18 EP disclosed