SCHEMBL8300989

SCHEMBL8300989

CN1CCC(c2cc3cccc(O)c3o2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
QDPR P09417 2/20 0.45
ACHE P22303 3/20 0.42
BCHE P06276 2/20 0.42
USP7 Q93009 1/20 0.40
PLG P00747 1/20 0.40
CDK1 P06493 1/20 0.40
CDK4 P11802 1/20 0.40
CCND1 P24385 1/20 0.40
CDK2 P24941 1/20 0.40
GSK3A P49840 1/20 0.40
GSK3B P49841 1/20 0.40
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM4 P08173 1/20 0.39
CHRM5 P08912 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29876097 0.86 MAOA (0.44) ACHEBCHEMAOAMAOB
SCHEMBL28792227 0.86 MAOA (0.44) ACHEBCHEMAOAMAOB
SCHEMBL8300351 0.82 SLC6A2 (0.59) QDPRACHEBCHESLC6A2SLC6A4
SCHEMBL8300839 0.79 ASAH1 (0.37) QDPRACHEBCHEPLGCDK1
SCHEMBL8290868 0.78 CHRM3 (0.41) CHRM3ASAH1
SCHEMBL9910974 0.77 ACHE (0.63) ACHEBCHESLC6A2SLC6A4CHRM2
SCHEMBL8300836 0.77 ASAH1 (0.45) ACHEBCHECHRM2CHRM4CHRM5
SCHEMBL8290869 0.77 ACHE (0.46) ACHEBCHESLC6A2SLC6A4CHRM2
Butane SCHEMBL8292425 0.75 USP2 (0.40) ACHEBCHESLC6A2SLC6A4ASAH1
SCHEMBL6603922 0.75 MAOA (0.38) ACHEBCHEMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0637586-B1 2-(Piperidin-4-yl, pyridin-4-yl and tetrahydropyridin-4-yl)-benzofuran-7-carbamate derivatives, their preparation and their use as acetylcholinesterase inhibitors HOECHST MARION ROUSSEL INC (US) 1999-06-02 EP disclosed
US-5708007-A ACETYLCHOLINESTERASE INHIBITORS HOECHST MARION ROUSSEL, INC. (US) 1998-01-13 US disclosed
EP-0637586-A1 2-(Piperidin-4-yl, pyridin-4-yl and tetrahydropyridin-4-yl)benzofuran-7-ol and carbamate derivatives, their preparation and their use as acetylcholinesterase inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1995-02-08 EP disclosed