SCHEMBL8300839

SCHEMBL8300839

CN1CCC(c2cc3cccc(N(C)C(=O)O)c3o2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ASAH1 Q13510 5/20 0.37
FAAH O00519 1/20 0.37
NAAA Q02083 1/20 0.37
CDK4 P11802 2/20 0.36
CCND1 P24385 2/20 0.36
CDK1 P06493 1/20 0.36
CDK2 P24941 1/20 0.36
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36
ACHE P22303 3/20 0.36
BCHE P06276 2/20 0.36
PLG P00747 1/20 0.36
KDM4E B2RXH2 1/20 0.35
QDPR P09417 1/20 0.35
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8300989 0.79 QDPR (0.45) ASAH1CDK4CCND1CDK1CDK2
SCHEMBL8292427 0.78 KDM4E (0.39) ASAH1FAAHNAAAACHEKDM4E
SCHEMBL8297441 0.76 ASAH1 (0.37) ASAH1FAAHNAAACDK4CCND1
SCHEMBL8300836 0.75 ASAH1 (0.45) ASAH1FAAHNAAAACHEBCHE
SCHEMBL8290868 0.74 CHRM3 (0.41) ASAH1KDM4ECHRM3CYP1A2
SCHEMBL8290869 0.73 ACHE (0.46) ASAH1ACHEBCHEKDM4ECHRM1
SCHEMBL8290905 0.73 BCHE (0.45) ACHEBCHEPLGKDM4EHTR2C
SCHEMBL8300351 0.73 SLC6A2 (0.59) ACHEBCHEKDM4EQDPRSLC6A2
SCHEMBL8292426 0.73 HPGD (0.42) ASAH1ACHEKDM4ESLC6A2SLC6A4
Butane SCHEMBL8292425 0.71 USP2 (0.40) ASAH1ACHEBCHEKDM4ESLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0637586-B1 2-(Piperidin-4-yl, pyridin-4-yl and tetrahydropyridin-4-yl)-benzofuran-7-carbamate derivatives, their preparation and their use as acetylcholinesterase inhibitors HOECHST MARION ROUSSEL INC (US) 1999-06-02 EP claimed