SCHEMBL8301109

SCHEMBL8301109

COc1ccc(C(=O)c2ccccc2C(=O)c2ccc3c(c2)OCO3)cc1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.61
NPC1 O15118 5/20 0.61
MAPT P10636 4/20 0.57
CTNNB1 P35222 3/20 0.57
WNT3A P56704 3/20 0.57
SMN1; SMN2 Q16637 3/20 0.57
ALDH1A1 P00352 2/20 0.56
LMNA P02545 1/20 0.56
HTT P42858 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
ALOX12 P18054 1/20 0.55
NFKB1 P19838 1/20 0.55
NFKB2 Q00653 1/20 0.55
RELA Q04206 1/20 0.55
SRD5A2 P31213 1/20 0.55
KMT2A Q03164 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.53
EDNRB P24530 1/20 0.53
EDNRA P25101 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4823544 0.90 RAB9A (0.68) RAB9ANPC1MAPTCTNNB1WNT3A
SCHEMBL5823399 0.84 CTNNB1 (0.57) RAB9ANPC1MAPTCTNNB1WNT3A
SCHEMBL4841835 0.84 SRD5A2 (0.56) RAB9ANPC1MAPTCTNNB1WNT3A
SCHEMBL7532873 0.83 SRD5A2 (0.69) RAB9ANPC1MAPTCTNNB1WNT3A
SCHEMBL4825307 0.81 RAB9A (0.64) RAB9ANPC1MAPTCTNNB1WNT3A
SCHEMBL4823371 0.81 CTNNB1 (0.78) RAB9ANPC1MAPTCTNNB1WNT3A
SCHEMBL4821161 0.80 CTNNB1 (0.61) RAB9ANPC1MAPTCTNNB1WNT3A
SCHEMBL15979976 0.78 CTNNB1 (0.78) RAB9ANPC1MAPTCTNNB1WNT3A
SCHEMBL26624014 0.78 KMT2A (0.72) RAB9ANPC1MAPTCTNNB1WNT3A
SCHEMBL1375270 0.78 KMT2A (0.68) RAB9ANPC1MAPTSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5929106-A VASODILATOR; HYPOTENSIVE AGENT SMITHKLINE BEECHAM CORPORATION (US) 1999-07-27 US disclosed
EP-0768878-A4 ENDOTHELIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-02-17 EP disclosed
US-5736564-A DIHYDROISOINDOLE DERIVATIVES SMITHKLINE BEECHAM CORPORATION (US) 1998-04-07 US disclosed
EP-0768878-A1 ENDOTHELIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-04-23 EP disclosed
WO-1995035107-A1 ENDOTHELIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1995-12-28 WO disclosed