SCHEMBL8301359

SCHEMBL8301359

COc1ccc2[nH]c(Cl)c(CC(=O)OCc3ccccc3)c2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.54
AKR1C2 P52895 1/20 0.51
MTNR1A P48039 5/20 0.48
MTNR1B P49286 5/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
MAPKAPK2 P49137 1/20 0.46
KDM4E B2RXH2 4/20 0.46
ALDH1A1 P00352 4/20 0.46
HSD17B10 Q99714 3/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ADORA2B P29275 1/20 0.46
HPGD P15428 2/20 0.46
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
MAPK1 P28482 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11014056 0.88 AKR1C2 (0.68) AKR1C2MTNR1AMTNR1BMEN1KMT2A
SCHEMBL19749132 0.84 AKR1C2 (0.48) AKR1C2MTNR1AMTNR1BMEN1KMT2A
SCHEMBL7962079 0.83 NQO2 (0.66) NQO2AKR1C2MTNR1AMTNR1BMEN1
SCHEMBL19749133 0.77 KDM4E (0.67) MTNR1AMTNR1BMEN1KMT2AKDM4E
SCHEMBL8301133 0.76 PLA2G2A (0.75) MEN1KMT2AALDH1A1CYP1A2CYP3A4
SCHEMBL11090385 0.74 MEN1 (0.53) NQO2AKR1C2MTNR1AMTNR1BMEN1
SCHEMBL28484096 0.73 TRPM8 (0.64) AKR1C2MEN1KMT2AKDM4EALDH1A1
SCHEMBL7964053 0.73 PLA2G2A (0.76) KMT2AMAPK1PTGS2PLA2G2A
SCHEMBL21336442 0.73 L3MBTL1 (0.65) MEN1KMT2AKDM4EALDH1A1HSD17B10
SCHEMBL5605077 0.72 AKR1C2 (0.74) NQO2AKR1C2MTNR1AMTNR1BMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620214-B1 1H-indole-3-acetic acid hydrazide sPLA2 inhibitors LILLY CO ELI (US) 1999-03-03 EP disclosed
US-5578634-A SEPTIC SHOCK TREATMENT ELI LILLY AND COMPANY (US) 1996-11-26 US disclosed
EP-0620214-A1 1H-indole-3-acetic acid hydrazide sPLA2 inhibitors ELI LILLY AND COMPANY (US) 1994-10-19 EP disclosed