SCHEMBL8301375

SCHEMBL8301375

CNS(=O)(=O)c1ccc(N)c(C(=O)NCc2ccc(OC)c(Cl)c2)c1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 2/20 0.53
GAA P10253 1/20 0.50
LMNA P02545 4/20 0.47
HPGD P15428 2/20 0.47
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8301665 0.87 NPC1 (0.52) GAALMNAHPGD
SCHEMBL8292287 0.84 GAA (0.57) NLRP3GAALMNAHPGD
SCHEMBL8299247 0.82 PDE5A (0.53) GAALMNAHPGD
SCHEMBL6944281 0.82 GAA (0.55) GAALMNAHPGD
SCHEMBL8299255 0.79 PDE5A (0.53) GAALMNAHPGD
SCHEMBL8416857 0.79 NLRP3 (0.45) NLRP3GAALMNAHPGDCYP1A2
SCHEMBL8416853 0.79 NLRP3 (0.45) NLRP3GAALMNAHPGDCYP1A2
SCHEMBL8297189 0.78 GAA (0.55) GAALMNAHPGDCYP1A2CYP2D6
SCHEMBL17241767 0.77 GAA (0.57) NLRP3GAALMNAHPGD
SCHEMBL8602155 0.76 POLB (0.49) NLRP3LMNACYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686625-B1 ANTHRANILIC ACID DERIVATIVE EISAI CO LTD (JP) 1999-05-26 EP disclosed
US-5716993-A PHOSPHODIESTERASE ENZYME INHIBITOR FOR TREATING CARDIOVASCULAR DISORDER, ANGINA PECTORIS, HYPERTENSION, ASTHMA EISAI CO., LTD. (JP) 1998-02-10 US disclosed
CN-1118595-A Anthranilic acid derivative EISAI CO LTD (JP) 1996-03-13 CN disclosed
EP-0686625-A1 ANTHRANILIC ACID DERIVATIVE Eisai Co., Ltd. (JP) 1995-12-13 EP disclosed