SCHEMBL8301453

SCHEMBL8301453

O=C(O)Oc1n[nH]cc1-c1cccc2ccccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.41
ADK P55263 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40
TDP1 Q9NUW8 2/20 0.39
PPARG P37231 5/20 0.38
PPARA Q07869 5/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
PPARD Q03181 1/20 0.38
MCL1 Q07820 1/20 0.38
ACMSD Q8TDX5 1/20 0.38
NR4A1 P22736 1/20 0.38
NR4A2 P43354 1/20 0.38
NR4A3 Q92570 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8297950 0.79 MEN1 (0.46) GSK3BADKMEN1KMT2AKDM4E
SCHEMBL10432295 0.78 ALDH1A1 (0.39) KDM4EALDH1A1TDP1HTTL3MBTL1
Hydrochloric Acid SCHEMBL27450739 0.78 MEN1 (0.44) GSK3BADKMEN1KMT2AKDM4E
SCHEMBL3391817 0.75 CDC7 (0.42) GSK3BADKMEN1KMT2AKDM4E
SCHEMBL2291368 0.74 ALDH1A1 (0.49) GSK3BADKMEN1KMT2AKDM4E
SCHEMBL1156690 0.73 ALDH1A1 (0.47) GSK3BADKMEN1KMT2AKDM4E
Bicarbonate SCHEMBL11569280 0.73 NR4A1 (0.58) MEN1KMT2AKDM4EALDH1A1HPGD
SCHEMBL11745392 0.73 DHFR (0.46) GSK3BMEN1KMT2AKDM4EALDH1A1
SCHEMBL6929782 0.72 MEN1 (0.51) MEN1KMT2AKDM4EALDH1A1HPGD
Bicarbonate SCHEMBL27535643 0.71 NR4A1 (0.56) MEN1KMT2AKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647629-B1 Neurotensin active substituted 1-naphthylpyrazole-3-carboxamides, their preparation and pharmaceutical compositions containing them SANOFI SA (FR) 1999-07-07 EP claimed