SCHEMBL8303069

SCHEMBL8303069

c1ccc(C(Oc2cccc3cc[nH]c23)(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 4/20 0.44
AHR P35869 2/20 0.42
KEAP1 Q14145 1/20 0.41
PDPK1 O15530 1/20 0.37
TRPA1 O75762 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
ITGB2 P05107 1/20 0.34
ICAM1 P05362 1/20 0.34
ITGAL P20701 1/20 0.34
CA4 P22748 1/20 0.34
CA6 P23280 1/20 0.34
ADK P55263 1/20 0.34
NR3C1 P04150 1/20 0.34
PGR P06401 1/20 0.34
NR3C2 P08235 1/20 0.34
AR P10275 1/20 0.34
BACE1 P56817 1/20 0.33
DRD4 P21917 1/20 0.32
HTR2A P28223 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL594299 0.77 BCHE (0.47) BCHEAHRKEAP1PDPK1TRPA1
SCHEMBL3789623 0.77 BCHE (0.51) BCHEAHRKEAP1PDPK1TRPA1
SCHEMBL4718619 0.74 KEAP1 (0.49) BCHEAHRKEAP1PDPK1TRPA1
SCHEMBL11064711 0.73 ALDH1A1 (0.54) PGRKDM4EALDH1A1HSD17B10MAPK1
SCHEMBL594125 0.71 BCHE (0.56) BCHEAHRKEAP1PDPK1CA1
SCHEMBL20049021 0.71 BCHE (0.51) BCHEAHRKEAP1PDPK1TRPA1
SCHEMBL28307887 0.71 BCHE (0.51) BCHEAHRKEAP1PDPK1TRPA1
SCHEMBL837602 0.70 L3MBTL1 (0.51) BCHEAHRMAPK1
SCHEMBL3870264 0.70 BCHE (0.48) BCHEAHRKEAP1PDPK1CA1
SCHEMBL5334267 0.70 BCHE (0.44) BCHEAHRKEAP1PDPK1TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0469833-B1 N-Benzyl-Indoles, processes for their preparation and pharmaceutical compositions containing them LILLY CO ELI (GB) 1999-09-08 EP disclosed
US-5281593-A Pharmaceuticals LILLY INDUSTRIES LIMITED (GB) 1994-01-25 US disclosed
EP-0469833-A1 N-Benzyl-Indoles, processes for their preparation and pharmaceutical compositions containing them LILLY INDUSTRIES LIMITED (GB) 1992-02-05 EP disclosed