SCHEMBL837602

SCHEMBL837602

c1ccc(COc2cccc3cc[nH]c23)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.51
MAPT P10636 1/20 0.51
MAPK1 P28482 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
LTA4H P09960 2/20 0.49
PLA2G2A P14555 1/20 0.49
TRPM8 Q7Z2W7 1/20 0.49
IDO1 P14902 1/20 0.47
HTR1A P08908 1/20 0.45
DRD2 P14416 1/20 0.45
BRD4 O60885 1/20 0.44
BCHE P06276 2/20 0.44
NSD2 O96028 1/20 0.44
ABL1 P00519 1/20 0.44
PPARG P37231 1/20 0.44
RIN1 Q13671 1/20 0.44
NCOR2 Q9Y618 1/20 0.44
LIPE Q05469 1/20 0.44
PTGER1 P34995 1/20 0.43
MAPK14 Q16539 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9023399 0.83 SRD5A2 (0.51) L3MBTL1MAPTMAPK1TDP1LTA4H
SCHEMBL23887763 0.78 LTA4H (0.54) L3MBTL1MAPTMAPK1TDP1LTA4H
SCHEMBL593890 0.77 BCHE (0.54) L3MBTL1MAPTBCHEPDE5AAHR
SCHEMBL7834454 0.77 POLB (0.43) L3MBTL1MAPTMAPK1TDP1HTR1A
Indole SCHEMBL28308979 0.77 DRD4 (0.56) L3MBTL1MAPTMAPK1TDP1HTR1A
SCHEMBL12313404 0.76 MAPT (0.47) L3MBTL1MAPTMAPK1TDP1LTA4H
SCHEMBL16632385 0.76 L3MBTL1 (0.44) L3MBTL1MAPTMAPK1TDP1IDO1
SCHEMBL30516781 0.75 KDM4E (0.57) L3MBTL1TDP1BCHEPOLBSMN1; SMN2
SCHEMBL4271654 0.75 MAPT (0.50) L3MBTL1MAPTMAPK1TDP1LTA4H
Charcoal, Activated SCHEMBL30421850 0.75 MAPT (0.46) L3MBTL1MAPTMAPK1TDP1LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 245 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112574093-B Novel green method for preparing 3-diaryl methyl substituted indole compound 湖南理工学院 2022-10-04 CN claimed
CN-112574093-A Novel green method for preparing 3-diaryl methyl substituted indole compound 湖南理工学院 2021-03-30 CN claimed
US-12599584-B2 Indoline derivatives, compositions comprising them and uses thereof YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM LTD. (IL) 2026-04-14 US disclosed
US-20250354000-A1 RUBBER COMPOSITION YOKOHAMA RUBBER CO LTD (JP) 2025-11-20 US disclosed
US-12473304-B2 Heterocyclic PAD4 inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2025-11-18 US disclosed
CN-115348961-B Heterocyclic PAD4 inhibitors 百时美施贵宝公司 2025-03-04 CN disclosed
US-20250059217-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF PREPARATION THEREOF BRIGHT MINDS BIOSCIENCES INC. (CA) 2025-02-20 US disclosed
CN-117897376-A Heterocyclic compounds and process for preparing same 光明智慧生物科学公司 2024-04-16 CN disclosed
EP-4347561-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF PREPARATION THEREOF Bright Minds Biosciences Inc. (CA) 2024-04-10 EP disclosed
US-11787783-B2 Heparanase inhibitors and use thereof Beta Therapeutics Pty Ltd (AU) 2023-10-17 US disclosed
US-11787783-B2 Heparanase inhibitors and use thereof Beta Therapeutics Pty Ltd (AU) 2023-10-17 US disclosed
EP-0548250-A4 SUBSTITUTED BICYCLIC ARYL COMPOUNDS EXHIBITING SELECTIVE LEUKOTRIENE B 4? ANTAGONIST ACTIVITY 1993-10-27 EP disclosed
EP-0548250-A1 SUBSTITUTED BICYCLIC ARYL COMPOUNDS EXHIBITING SELECTIVE LEUKOTRIENE B 4? ANTAGONIST ACTIVITY. RHONE POULENC RORER INT (US) 1993-06-30 EP disclosed
WO-1993001813-A1 PLATELET ACTIVATING FACTOR ANTAGONISTS ABBOTT LABORATORIES (US) 1993-02-04 WO disclosed
WO-1992014732-A1 INDOLES USEFUL AS PLATELET ACTIVATING FACTOR ANTAGONISTS ABBOTT LABORATORIES (US) 1992-09-03 WO disclosed
EP-0499987-A1 Platelet activating factor antagonists ABBOTT LABORATORIES (US) 1992-08-26 EP disclosed
CN-1061413-A Medicinal compound LILLY INDUSTRIES LTD (GB) 1992-05-27 CN disclosed
WO-1992004321-A1 SUBSTITUTED BICYCLIC ARYL COMPOUNDS EXHIBITING SELECTIVE LEUKOTRIENE B4 ANTAGONIST ACTIVITY RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1992-03-19 WO disclosed
EP-0469833-A1 N-Benzyl-Indoles, processes for their preparation and pharmaceutical compositions containing them LILLY INDUSTRIES LIMITED (GB) 1992-02-05 EP disclosed
US-4810699-A Substituted 1,3,4,9-tetrahydropyrano[3,4,-b]indole-1-acetic acids, pharmaceutical compositions containing them, and methods for treating inflammatory conditions and for analgesic purposes using them AMERICAN HOME PRODUCTS CORPORATION (US) 1989-03-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12473304-B2 Heterocyclic PAD4 inhibitors PADI6, PADI4, PADI1 L3MBTL1 1757/4885MAPT 4383/4885MAPK1 2514/4885
US-20250059217-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF PREPARATION THEREOF OPRL1, OPRK1, CNR2 L3MBTL1 4682/4885MAPT 435/4885MAPK1 158/4885
US-11787783-B2 Heparanase inhibitors and use thereof HPSE, HEXD, ENGASE L3MBTL1 4413/4885MAPT 2923/4885MAPK1 2482/4885
US-12599584-B2 Indoline derivatives, compositions comprising them and uses thereof IL6, TNF, IDO1 L3MBTL1 1914/4885MAPT 2305/4885MAPK1 1443/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.