SCHEMBL8303311

SCHEMBL8303311

CCS(=O)(=O)N(C)c1cccc(C(=O)O)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.46
LMNA P02545 2/20 0.46
ALDH1A1 P00352 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.45
NSD2 O96028 1/20 0.45
ESR1 P03372 1/20 0.45
POLB P06746 1/20 0.45
APEX1 P27695 1/20 0.45
RECQL P46063 1/20 0.45
ESR2 Q92731 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
GRM2 Q14416 2/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA6 P23280 1/20 0.42
CA9 Q16790 1/20 0.42
LTB4R2 Q9NPC1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30006467 0.83 LMNA (0.51) KMT2ALMNAALDH1A1L3MBTL1HTT
SCHEMBL3855094 0.83 LMNA (0.51) KMT2ALMNAALDH1A1L3MBTL1HTT
SCHEMBL14536599 0.83 POLB (0.49) KMT2AALDH1A1L3MBTL1POLBHTT
SCHEMBL5928422 0.83 ALDH1A1 (0.48) KMT2ALMNAALDH1A1L3MBTL1NSD2
SCHEMBL6246429 0.82 AKR1C3 (0.48) KMT2ALMNAALDH1A1L3MBTL1PPARA
SCHEMBL6244788 0.81 L3MBTL1 (0.43) KMT2ALMNAALDH1A1L3MBTL1NSD2
SCHEMBL5529874 0.80 MAPT (0.56) KMT2ALMNAALDH1A1L3MBTL1POLB
SCHEMBL4702681 0.80 MAPT (0.56) KMT2ALMNAALDH1A1L3MBTL1POLB
SCHEMBL6417389 0.79 LMNA (0.62) KMT2ALMNAALDH1A1HTTSMN1; SMN2
SCHEMBL6273186 0.79 ESR1 (0.50) KMT2ALMNAALDH1A1L3MBTL1NSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005009995-A1 NICOTINAMIDE DERIVATIVES USEFUL AS PDE4 INHIBITORS PFIZER LIMITED (GB) 2005-02-03 WO disclosed