SCHEMBL8303701

SCHEMBL8303701

CCOC(=O)CC(=O)c1ccc(C#N)cc1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.48
NPSR1 Q6W5P4 1/20 0.48
MAP2K1 Q02750 3/20 0.44
KMT2A Q03164 4/20 0.43
MEN1 O00255 3/20 0.43
MIF P14174 1/20 0.43
PDCD1 Q15116 1/20 0.41
CD274 Q9NZQ7 1/20 0.41
TP53 P04637 1/20 0.41
THRB P10828 1/20 0.41
MAPT P10636 3/20 0.40
POLB P06746 1/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
PKM P14618 1/20 0.40
GPR27 Q9NS67 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5869086 0.89 MIF (0.43) GAANPSR1MAP2K1KMT2AMEN1
SCHEMBL7887305 0.86 MIF (0.40) GAANPSR1MAP2K1KMT2AMEN1
SCHEMBL1823015 0.86 MIF (0.44) GAANPSR1MAP2K1KMT2AMEN1
SCHEMBL4178450 0.84 CA12 (0.47) GAANPSR1MAP2K1KMT2AMEN1
SCHEMBL7889566 0.82 GABRA1 (0.43) GAANPSR1KMT2AMEN1MIF
SCHEMBL2080446 0.81 CES2 (0.49) GAANPSR1KMT2AMEN1MIF
SCHEMBL12692656 0.81 NLRP3 (0.44) GAANPSR1KMT2AMEN1MIF
SCHEMBL406494 0.81 GAA (0.49) GAANPSR1MAP2K1KMT2AMEN1
SCHEMBL13537990 0.79 MIF (0.42) GAANPSR1KMT2AMEN1MIF
SCHEMBL1568667 0.79 DGAT1 (0.49) GAANPSR1MAP2K1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0906285-A1 3-CYANOARYL PYRAZOLES AND USE THEREOF AS HERBICIDES BAYER AG (DE) 1999-04-07 EP disclosed
WO-1997046535-A1 3-CYANOARYL PYRAZOLES AND USE THEREOF AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 1997-12-11 WO disclosed
WO-1996001255-A1 3-(CYANOPHENYL)-PYRAZOLE DERIVATIVES AS HERBICIDES ZENECA LIMITED (GB) 1996-01-18 WO disclosed