SCHEMBL8303909

SCHEMBL8303909

CCC(N)c1ccc([Si](C)(C)C)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.53
CYP1A2 P05177 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C19 P33261 2/20 0.33
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32
SLC2A1 P11166 1/20 0.32
ROCK1 Q13464 1/20 0.31
TDP1 Q9NUW8 2/20 0.31
LMNA P02545 1/20 0.31
ESR1 P03372 1/20 0.31
PGR P06401 1/20 0.31
CHRM2 P08172 1/20 0.31
CYP3A4 P08684 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
AR P10275 1/20 0.31
MAPT P10636 1/20 0.31
CHRM1 P11229 1/20 0.31
CYP2C9 P11712 1/20 0.31
ALOX15 P16050 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23092069 0.83 SLC6A4 (0.70) SLC6A4CYP1A2CYP2D6CYP2C19SLC2A1
SCHEMBL14648925 0.76 ALDH1A1 (0.42) CYP1A2CYP2D6CYP2C19TDP1MAPT
SCHEMBL3863807 0.75 SLC6A4 (0.59) SLC6A4CYP1A2CYP2D6CYP2C19TDP1
SCHEMBL8305051 0.75 ADRB2 (0.52) NR1H2NR1H3ROCK1
SCHEMBL8284225 0.75 SLC6A4 (0.59) SLC6A4CYP1A2CYP2D6CYP2C19TDP1
SCHEMBL8286101 0.75 SLC6A4 (0.59) SLC6A4CYP1A2CYP2D6CYP2C19TDP1
SCHEMBL238408 0.75 SLC6A4 (0.59) SLC6A4CYP1A2CYP2D6CYP2C19SLC2A1
SCHEMBL8285910 0.75 SLC6A4 (0.59) SLC6A4CYP1A2CYP2D6CYP2C19TDP1
SCHEMBL3865060 0.75 SLC6A4 (0.59) SLC6A4CYP1A2CYP2D6CYP2C19TDP1
SCHEMBL6193234 0.73 SLC6A4 (0.57) SLC6A4CYP1A2CYP2D6CYP2C19SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0555388-B1 INSECTICIDAL, ACARICIDAL AND FUNGICIDAL AMINOPYRIMIDINES DU PONT (US) 1999-01-27 EP disclosed
US-5378708-A Agricultural pesticides E. I. DU PONT DE NEMOURS AND COMPANY (US) 1995-01-03 US disclosed
EP-0555388-A1 INSECTICIDAL, ACARICIDAL AND FUNGICIDAL AMINOPYRIMIDINES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1993-08-18 EP disclosed
WO-1992008704-A1 INSECTICIDAL, ACARICIDAL AND FUNGICIDAL AMINOPYRIMIDINES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1992-05-29 WO disclosed