SCHEMBL8305051

SCHEMBL8305051

CC(N)c1ccc([Si](C)(C)C)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.52
PDE2A O00408 1/20 0.47
ROCK2 O75116 5/20 0.37
ROCK1 Q13464 3/20 0.37
NR1H2 P55055 2/20 0.35
NR1H3 Q13133 2/20 0.35
CIT O14578 2/20 0.35
PRKD3 O94806 1/20 0.33
MAP4K4 O95819 1/20 0.33
PRKCB P05771 1/20 0.33
PRKCA P17252 1/20 0.33
PRKACA P17612 1/20 0.33
CSNK2A2 P19784 1/20 0.33
MARK3 P27448 1/20 0.33
BMPR1A P36894 1/20 0.33
CSNK1A1 P48729 1/20 0.33
CLK1 P49759 1/20 0.33
GSK3A P49840 1/20 0.33
GSK3B P49841 1/20 0.33
CDK9 P50750 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1314596 0.81 ADRB2 (0.72) ADRB2PDE2AROCK2ROCK1CIT
SCHEMBL6124152 0.79 TYR (0.42) NR1H2NR1H3
SCHEMBL15259491 0.78 ADRB2 (0.56) ADRB2PDE2AROCK2ROCK1CIT
SCHEMBL28646449 0.75 ALDH1A1 (0.42) NR1H2NR1H3GSK3B
SCHEMBL8308999 0.75 NR1H2 (0.35) NR1H2NR1H3
SCHEMBL8737598 0.75 NR1H2 (0.35) NR1H2NR1H3
SCHEMBL8303909 0.75 SLC6A4 (0.53) ROCK1NR1H2NR1H3
SCHEMBL14980120 0.75 ABCB11 (0.42) NR1H2NR1H3
SCHEMBL586534 0.74 NR1H2 (0.50) NR1H2NR1H3
SCHEMBL25077966 0.73 ACHE (0.37) ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0555388-B1 INSECTICIDAL, ACARICIDAL AND FUNGICIDAL AMINOPYRIMIDINES DU PONT (US) 1999-01-27 EP disclosed
US-5378708-A Agricultural pesticides E. I. DU PONT DE NEMOURS AND COMPANY (US) 1995-01-03 US disclosed
WO-1993022291-A1 ARTHROPODICIDAL AND FUNGICIDAL AMINOPYRIMIDINES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1993-11-11 WO disclosed
EP-0555388-A1 INSECTICIDAL, ACARICIDAL AND FUNGICIDAL AMINOPYRIMIDINES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1993-08-18 EP disclosed
WO-1992008704-A1 INSECTICIDAL, ACARICIDAL AND FUNGICIDAL AMINOPYRIMIDINES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1992-05-29 WO disclosed