SCHEMBL8303940

SCHEMBL8303940

NC(=O)C1CCN(c2ccccc2)C(=O)C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.49
NPSR1 Q6W5P4 2/20 0.49
KDM4E B2RXH2 1/20 0.49
SMN1; SMN2 Q16637 4/20 0.48
PKM P14618 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
CYP2C19 P33261 1/20 0.46
USP30 Q70CQ3 2/20 0.45
RAB9A P51151 2/20 0.45
TSHR P16473 2/20 0.45
NPC1 O15118 2/20 0.45
MEN1 O00255 1/20 0.45
TDP2 O95551 1/20 0.45
POLB P06746 1/20 0.45
HPGD P15428 1/20 0.45
CASP3 P42574 1/20 0.45
GALK1 P51570 1/20 0.45
KMT2A Q03164 1/20 0.45
ATM Q13315 1/20 0.45
HKDC1 Q2TB90 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8305161 0.87 NOTUM (0.54) ALDH1A1SMN1; SMN2USP30TSHRNPC1
SCHEMBL16131376 0.84 RAB9A (0.60) ALDH1A1SMN1; SMN2RAB9ATSHRNPC1
SCHEMBL8305710 0.81 ALDH1A1 (0.51) ALDH1A1NPSR1SMN1; SMN2USP30RAB9A
SCHEMBL3529467 0.78 NOTUM (0.64) ALDH1A1NPSR1KDM4ESMN1; SMN2PKM
SCHEMBL1661083 0.77 NPC1 (0.60) ALDH1A1NPSR1KDM4EPKMTSHR
Benzene SCHEMBL28217786 0.77 NOTUM (0.62) ALDH1A1NPSR1KDM4ESMN1; SMN2PKM
Hydrochloric Acid SCHEMBL28060567 0.77 NOTUM (0.62) ALDH1A1NPSR1KDM4ESMN1; SMN2PKM
SCHEMBL5104476 0.74 USP30 (0.51) ALDH1A1NPSR1KDM4EUSP30RAB9A
SCHEMBL5326027 0.74 ITGB3 (0.45) ALDH1A1KDM4ECYP2C19TSHRPOLB
Cadaverine Tartrate SCHEMBL29195643 0.74 POLB (0.40) ALDH1A1SMN1; SMN2USP30RAB9ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965578-A Inhibitors of farnesyl-protein transferase MERCK & CO., INC. (US) 1999-10-12 US disclosed
EP-0897303-A4 1999-02-24 EP disclosed
EP-0897303-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1999-02-24 EP disclosed
WO-1997036605-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1997-10-09 WO disclosed