SCHEMBL8304320

SCHEMBL8304320

CN(Cc1ccccc1)C(=O)c1ccc2c(NCc3cccc(C(=N)N)c3)ncnc2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
CYP1A2 P05177 3/20 0.49
CYP3A4 P08684 3/20 0.49
MAPK1 P28482 3/20 0.49
CYP2C19 P33261 3/20 0.49
HSD17B10 Q99714 3/20 0.49
USP2 O75604 2/20 0.49
LMNA P02545 2/20 0.49
CYP2D6 P10635 2/20 0.49
CLK4 Q9HAZ1 1/20 0.49
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
F10 P00742 1/20 0.47
KDM4E B2RXH2 2/20 0.47
HPGD P15428 2/20 0.47
CYP2C9 P11712 1/20 0.47
ALOX12 P18054 1/20 0.47
RPS6KB1 P23443 5/20 0.46
AURKA O14965 5/20 0.46
AURKB Q96GD4 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6324691 0.86 AURKA (0.48) ALDH1A1CYP1A2CYP3A4MAPK1CYP2C19
SCHEMBL6327136 0.83 POLB (0.46) ALDH1A1CYP1A2CYP3A4MAPK1CYP2C19
SCHEMBL6329487 0.79 AURKA (0.43) ALDH1A1CYP1A2CYP3A4MAPK1CYP2C19
SCHEMBL6329960 0.79 F10 (0.48) MAPK1F10RPS6KB1AURKAAURKB
SCHEMBL8307208 0.78 F10 (0.48) LMNAF10HPGDRPS6KB1AURKA
SCHEMBL6325892 0.78 F10 (0.48) LMNAF10HPGDRPS6KB1AURKA
Hydrochloric Acid SCHEMBL6326766 0.78 F10 (0.48) MAPK1F10RPS6KB1AURKAAURKB
Hydrochloric Acid SCHEMBL6325502 0.78 F10 (0.47) LMNAF10HPGDRPS6KB1AURKA
SCHEMBL6322361 0.78 AURKA (0.49) LMNAF10HPGDRPS6KB1AURKA
SCHEMBL6323882 0.74 MEN1 (0.56) ALDH1A1MEN1KMT2AHPGDADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004080970-A1 NOVEL BICYCLIC AROMATIC COMPOUNDS, THE PRODUCTION AND USE THEREOF IN THE FORM OF DRUGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2004-09-23 WO disclosed