SCHEMBL8304375

SCHEMBL8304375

NC(c1ccncc1)C1CCN(C2CCC(CC(=O)O)CC2)CC1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.43
ITGA2B P08514 2/20 0.43
KDM4E B2RXH2 3/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KMT2A Q03164 1/20 0.39
TRPV6 Q9H1D0 2/20 0.38
HTR2A P28223 1/20 0.38
HRH1 P35367 1/20 0.38
HTR2B P41595 1/20 0.38
RECQL P46063 1/20 0.37
CCNT1 O60563 2/20 0.36
CDK9 P50750 2/20 0.36
ANPEP P15144 1/20 0.35
ENPEP Q07075 1/20 0.35
ROCK2 O75116 2/20 0.35
FFAR4 Q5NUL3 3/20 0.34
DGAT1 O75907 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8300200 0.81 KDM4E (0.37) ITGB3ITGA2BKDM4EMEN1ALDH1A1
SCHEMBL8613755 0.76 ITGB3 (0.56) ITGB3ITGA2BKDM4EMEN1ALDH1A1
SCHEMBL8301327 0.76 KDM4E (0.43) ITGB3ITGA2BKDM4EMEN1ALDH1A1
SCHEMBL8298757 0.76 HRH3 (0.49) ITGB3ITGA2BFFAR4
SCHEMBL8300331 0.73 KDM4E (0.43) ITGB3ITGA2BKDM4EMEN1ALDH1A1
SCHEMBL8305336 0.73 KDM4E (0.43) ITGB3ITGA2BKDM4EMEN1ALDH1A1
SCHEMBL8298652 0.73 ITGB3 (0.45) ITGB3ITGA2BKDM4EMEN1ALDH1A1
SCHEMBL16499811 0.71 HTR2A (0.44) ITGB3ITGA2BKDM4EALDH1A1HTR2A
SCHEMBL8300686 0.70 NAMPT (0.43) ITGB3ITGA2BKDM4EMEN1ALDH1A1
SCHEMBL8300030 0.70 KDM4E (0.45) ITGB3ITGA2BKDM4EMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808306-B1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 1999-08-04 EP disclosed