SCHEMBL8300200

SCHEMBL8300200

NC(c1ccncc1)C1CCN(C2CCC(O)(CC(=O)O)CC2)CC1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
KMT2A Q03164 1/20 0.37
ITGB3 P05106 7/20 0.34
ITGA2B P08514 7/20 0.34
HRH3 Q9Y5N1 3/20 0.34
TRPV6 Q9H1D0 1/20 0.34
RECQL P46063 1/20 0.33
OPRL1 P41146 1/20 0.33
DPP4 P27487 1/20 0.32
DPP8 Q6V1X1 1/20 0.32
DPP9 Q86TI2 1/20 0.32
DPP7 Q9UHL4 1/20 0.32
HTR2A P28223 1/20 0.32
HRH1 P35367 1/20 0.32
HTR2B P41595 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8304375 0.81 ITGB3 (0.43) KDM4EMEN1ALDH1A1KMT2AITGB3
SCHEMBL7399380 0.78 ITGB3 (0.49) KDM4EMEN1ALDH1A1KMT2AITGB3
SCHEMBL7399382 0.78 ITGB3 (0.49) KDM4EMEN1ALDH1A1KMT2AITGB3
SCHEMBL8303817 0.77 KDM4E (0.40) KDM4EMEN1ALDH1A1KMT2AITGB3
SCHEMBL8300631 0.74 GRIN2B (0.40) KDM4EMEN1ALDH1A1KMT2AITGB3
SCHEMBL8301361 0.72 CYP2D6 (0.39) KDM4EMEN1ALDH1A1KMT2AITGB3
SCHEMBL8300676 0.72 KDM4E (0.42) KDM4EMEN1ALDH1A1KMT2AITGB3
SCHEMBL8299936 0.70 KDM4E (0.41) KDM4EMEN1ALDH1A1KMT2ATRPV6
SCHEMBL8615320 0.70 KDM2B (0.34) KDM4EMEN1ALDH1A1KMT2AITGB3
SCHEMBL8301126 0.70 KDM4E (0.40) KDM4EMEN1ALDH1A1KMT2ATRPV6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808306-B1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 1999-08-04 EP disclosed