SCHEMBL8306288

SCHEMBL8306288

Cc1cccc(-c2cc3ccccc3[nH]2)c1-c1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 1/20 0.55
ATM Q13315 1/20 0.55
ATR Q13535 1/20 0.55
CA12 O43570 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA9 Q16790 1/20 0.54
PTGS2 P35354 9/20 0.47
CNR1 P21554 1/20 0.46
KDR P35968 2/20 0.46
AURKA O14965 1/20 0.46
KDM4E B2RXH2 2/20 0.45
MEN1 O00255 2/20 0.45
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45
HPGD P15428 2/20 0.45
KMT2A Q03164 2/20 0.45
USP2 O75604 1/20 0.45
LMNA P02545 1/20 0.45
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8307211 0.85 CA12 (0.57) PRKDCATMATRCA12CA1
SCHEMBL8305443 0.82 CA12 (0.72) PRKDCATMATRCA12CA1
SCHEMBL3433722 0.81 KDM4E (0.55) CA12CA1CA2CA9KDR
SCHEMBL8307758 0.81 PRKDC (0.55) PRKDCATMATRCA12CA1
SCHEMBL8521718 0.80 KDM4E (0.58) PRKDCATMATRCA12CA1
SCHEMBL29941586 0.74 RAB9A (0.62) KDRAURKAKDM4EMEN1ALDH1A1
SCHEMBL4890695 0.74 RAB9A (0.62) KDRAURKAKDM4EMEN1ALDH1A1
SCHEMBL30292823 0.73 PTGS2 (0.60) PRKDCATMATRCA12CA1
SCHEMBL29727516 0.73 KDR (0.60) CA12CA1CA2CA9KDR
SCHEMBL517386 0.71 CA1 (0.52) CA12CA1CA2CA9PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915848-A1 1,2-DIARYLINDOLE AS COX-2 INHIBITORS LABORATOIRES UPSA (FR) 1999-05-19 EP disclosed
WO-1998005639-A1 1,2-DIARYLINDOLE AS COX-2 INHIBITORS LABORATOIRES UPSA (FR) 1998-02-12 WO disclosed