SCHEMBL8307758

SCHEMBL8307758

CS(=O)(=O)c1ccc(-c2ccc(S(C)(=O)=O)cc2-c2cc3ccccc3[nH]2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 1/20 0.55
ATM Q13315 1/20 0.55
ATR Q13535 1/20 0.55
CA12 O43570 1/20 0.55
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
CA9 Q16790 1/20 0.55
PTGS2 P35354 10/20 0.52
CNR1 P21554 1/20 0.49
CHEK1 O14757 1/20 0.47
KDR P35968 1/20 0.47
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
USP2 O75604 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
POLB P06746 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8307211 0.92 CA12 (0.57) PRKDCATMATRCA12CA1
SCHEMBL8521718 0.91 KDM4E (0.58) PRKDCATMATRCA12CA1
SCHEMBL8305443 0.86 CA12 (0.72) PRKDCATMATRCA12CA1
SCHEMBL8306288 0.81 PRKDC (0.55) PRKDCATMATRCA12CA1
SCHEMBL30292823 0.79 PTGS2 (0.60) PRKDCATMATRCA12CA1
SCHEMBL25726938 0.79 PTGS2 (0.50) PRKDCATMATRCA12CA1
SCHEMBL8306238 0.75 CDK5 (0.60) PRKDCATMATRCA12CA1
SCHEMBL28929657 0.73 CA2 (0.77) PRKDCATMATRCA12CA1
SCHEMBL25727641 0.72 CYP19A1 (0.55) PRKDCATMATRCA12CA1
SCHEMBL10997079 0.71 RAB9A (0.71) CA12CA1CA2CA9CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915848-A1 1,2-DIARYLINDOLE AS COX-2 INHIBITORS LABORATOIRES UPSA (FR) 1999-05-19 EP disclosed
WO-1998005639-A1 1,2-DIARYLINDOLE AS COX-2 INHIBITORS LABORATOIRES UPSA (FR) 1998-02-12 WO disclosed