SCHEMBL8306437

SCHEMBL8306437

COC(=O)/C=C(/Cc1cc(F)c(F)cc1F)N[C@H](C(N)=O)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.38
GPR88 Q9GZN0 1/20 0.36
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.35
NR1H3 Q13133 1/20 0.35
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
ALDH1A1 P00352 2/20 0.34
TACR3 P29371 1/20 0.34
ATM Q13315 1/20 0.33
RORC P51449 1/20 0.33
GAA P10253 1/20 0.33
SYK P43405 1/20 0.33
CNR2 P34972 1/20 0.33
ANPEP P15144 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8302507 0.83 CNR2 (0.44) GPR88KMT2AMEN1CYP3A4CYP2D6
SCHEMBL14688086 0.78 CYP3A4 (0.47) KMT2AMEN1CYP3A4CYP2D6CYP2C9
SCHEMBL14688085 0.78 CYP3A4 (0.47) KMT2AMEN1CYP3A4CYP2D6CYP2C9
SCHEMBL18683717 0.76 CYP3A4 (0.41) KMT2AMEN1CYP3A4CYP2D6CYP2C9
SCHEMBL14701601 0.76 CYP3A4 (0.41) KMT2AMEN1CYP3A4CYP2D6CYP2C9
SCHEMBL31011124 0.76 ALDH1A1 (0.41) KMT2AMEN1CYP2D6CYP2C9CYP2C19
SCHEMBL29172249 0.76 KMT2A (0.42) DPP4KMT2AMEN1CYP3A4CYP2D6
SCHEMBL8307199 0.73 TSHR (0.43) GPR88KMT2ACYP3A4CYP2C9ALDH1A1
SCHEMBL13780954 0.73 DPP4 (0.36) DPP4RORC
SCHEMBL2861837 0.73 DPP4 (0.41) DPP4CYP2D6RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004085661-A2 PROCESS TO CHIRAL BETA-AMINO ACID DERIVATIVES MERCK & CO., INC (US) 2004-10-07 WO disclosed