SCHEMBL8302507

SCHEMBL8302507

COC(=O)/C=C(/Cc1ccccc1)N[C@H](C(N)=O)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 7/20 0.44
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.41
CYP3A4 P08684 1/20 0.41
GAA P10253 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41
ATM Q13315 1/20 0.40
CNR1 P21554 1/20 0.40
GPR88 Q9GZN0 1/20 0.40
ALDH1A1 P00352 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
EPHX1 P07099 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8303023 0.87 CNR2 (0.49) CNR2KMT2ACNR1ALDH1A1MAPT
SCHEMBL8306437 0.83 DPP4 (0.38) CNR2MEN1KMT2ACYP3A4GAA
SCHEMBL8307199 0.80 TSHR (0.43) KMT2APOLBCYP3A4CYP2C9TSHR
SCHEMBL8302401 0.77 GPR88 (0.40) KMT2ACYP1A2POLBCYP3A4GAA
SCHEMBL4566800 0.77 CNR2 (0.67) CNR2MEN1KMT2APOLBCNR1
SCHEMBL8305615 0.77 CNR2 (0.46) CNR2MEN1KMT2AGAATSHR
SCHEMBL9003082 0.74 ALDH1A1 (0.46) CNR2MEN1KMT2ACYP1A2CYP3A4
SCHEMBL9003077 0.74 ALDH1A1 (0.46) CNR2MEN1KMT2ACYP1A2CYP3A4
SCHEMBL8303022 0.73 ALDH1A1 (0.46) MEN1KMT2APOLBCYP3A4GAA
SCHEMBL18653054 0.73 CYP2D6 (0.51) KMT2ACYP3A4CYP2D6CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004085661-A2 PROCESS TO CHIRAL BETA-AMINO ACID DERIVATIVES MERCK & CO., INC (US) 2004-10-07 WO disclosed