SCHEMBL8306828

SCHEMBL8306828

Cc1ccsc1Cc1ccc(F)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
HPGD P15428 2/20 0.47
LMNA P02545 1/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
PKM P14618 1/20 0.47
ADRA1D P25100 2/20 0.44
POLB P06746 1/20 0.39
TAAR1 Q96RJ0 1/20 0.38
PTGS1 P23219 2/20 0.38
PTGS2 P35354 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
ALOX5 P09917 1/20 0.38
RAB9A P51151 2/20 0.37
NPC1 O15118 1/20 0.37
TP53 P04637 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
IDO1 P14902 1/20 0.35
LOXL2 Q9Y4K0 1/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6947065 0.80 ADRA1D (0.46) ALDH1A1HPGDLMNAGAAMAPT
Ethylamine SCHEMBL10586929 0.74 ADRA1D (0.39) ALDH1A1HPGDLMNAADRA1DSMN1; SMN2
SCHEMBL8304165 0.73 MAPT (0.40) ALDH1A1HPGDLMNAGAAMAPT
SCHEMBL10445253 0.72
SCHEMBL2976063 0.72 PTGS1 (0.41) ALDH1A1HPGDLMNAGAAMAPT
SCHEMBL1468357 0.68 IDO1 (0.58) ALDH1A1LMNATAAR1IDO1LOXL2
SCHEMBL16561361 0.68 IDO1 (0.58) ALDH1A1LMNATAAR1IDO1LOXL2
SCHEMBL12425696 0.68 TAAR1 (0.45) ALDH1A1ADRA1DTAAR1NPC1IDO1
SCHEMBL256017 0.68
SCHEMBL3689463 0.68 ACHE (0.68) ALDH1A1HPGDLMNAGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0667855-B1 SUBSTITUTED ARYLALKYNYL- AND HETEROARYLALKYNYL-N-HYDROXYUREA INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS ABBOTT LAB (US) 1999-03-24 EP disclosed
US-5616596-A Substituted arylalkynyl-and heteroarylalkynl-N-hydroxyurea inhibitors of leukotriene biosynthesis ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
EP-0667855-A4 SUBSTITUTED ARYLALKYNYL- AND HETEROARYLALKYNYL-N-HYDROXYUREA INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS. ABBOTT LAB (US) 1996-02-21 EP disclosed
EP-0667855-A1 SUBSTITUTED ARYLALKYNYL- AND HETEROARYLALKYNYL-N-HYDROXYUREA INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS ABBOTT LABORATORIES (US) 1995-08-23 EP disclosed
WO-1994011342-A1 SUBSTITUTED ARYLALKYNYL- AND HETEROARYLALKYNYL-N-HYDROXYUREA INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS ABBOTT LABORATORIES (US) 1994-05-26 WO disclosed