SCHEMBL8307047

SCHEMBL8307047

O=C1Nc2ccc(S(=O)(=O)N3CCC[C@@H]3CO)cc2C1(Cl)Cl

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 16/20 0.49
CASP7 P55210 12/20 0.49
CASP9 P55211 3/20 0.49
CASP1 P29466 7/20 0.48
GAA P10253 1/20 0.48
PLAU P00749 1/20 0.47
CASP6 P55212 4/20 0.46
CASP2 P42575 3/20 0.46
CASP4 P49662 2/20 0.46
CASP8 Q14790 2/20 0.46
LOX P28300 1/20 0.45
BRD4 O60885 1/20 0.44
BRD2 P25440 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6954700 1.00 CASP3 (0.49) CASP3CASP7CASP9CASP1GAA
SCHEMBL7440426 0.88 CASP3 (0.51) CASP3CASP7CASP9CASP1GAA
SCHEMBL8307728 0.86 CASP3 (0.68) CASP3CASP7CASP9CASP1
SCHEMBL6947728 0.86 CASP3 (0.68) CASP3CASP7CASP9CASP1
SCHEMBL7444177 0.81 CYP3A4 (0.57) CASP3CASP7CASP9CASP1GAA
SCHEMBL6535733 0.80 CASP3 (0.74) CASP3CASP7CASP9CASP1CASP6
SCHEMBL7433422 0.80 PSEN1 (0.56) CASP3CASP7CASP9GAA
SCHEMBL6535888 0.80 CASP3 (0.74) CASP3CASP7CASP9CASP1CASP6
SCHEMBL6951145 0.77 FKBP1A (0.58) CASP3CASP7GAA
SCHEMBL6954598 0.76 GAA (0.63) CASP3CASP7CASP9CASP1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004078731-A1 QUINOLINE-CARBOXYLIC ACIDS AND THE DERIVATIVES THEREOF, A FOCUSED LIBRARY 'CHEMICAL DIVERSITY RESEARCH INSTITUTE', LTD. (RU) 2004-09-16 WO disclosed