SCHEMBL8307403

SCHEMBL8307403

NC(=O)N1CCNCC1.O=C(O)c1c[nH]c2ccccc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.55
ATM Q13315 1/20 0.55
HTR3E A5X5Y0 1/20 0.52
HTR3B O95264 1/20 0.52
HTR3A P46098 1/20 0.52
HTR3D Q70Z44 1/20 0.52
HTR3C Q8WXA8 1/20 0.52
GFER P55789 1/20 0.52
POLB P06746 1/20 0.51
GPR84 Q9NQS5 1/20 0.50
LMNA P02545 2/20 0.49
HTT P42858 1/20 0.49
MAPK14 Q16539 1/20 0.49
KDM4E B2RXH2 1/20 0.49
GABRA1 P14867 2/20 0.48
GABRG2 P18507 2/20 0.48
GABRB3 P28472 2/20 0.48
GABRA3 P34903 2/20 0.48
GABRA2 P47869 2/20 0.48
GABRB2 P47870 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3380253 0.88 POLB (0.67) ALDH1A1ATMGFERPOLBGPR84
Piperazine SCHEMBL7073764 0.84 HTR3E (0.65) ALDH1A1ATMHTR3EHTR3BHTR3A
SCHEMBL1144650 0.83 GFER (0.68) ALDH1A1ATMHTR3EHTR3BHTR3A
SCHEMBL3994500 0.81 POLB (0.77) ALDH1A1HTR3EHTR3BHTR3AHTR3D
Piperidine SCHEMBL8707735 0.80 HTR3E (0.60) ALDH1A1ATMHTR3EHTR3BHTR3A
Hydrazine SCHEMBL27559974 0.79 ALDH1A1 (0.72) ALDH1A1ATMGPR84KDM4EGABRA1
SCHEMBL64182 0.79 GPR84 (0.77) ALDH1A1ATMGPR84KDM4EGABRA1
SCHEMBL3449612 0.77 HTR3E (0.51) ALDH1A1ATMHTR3EHTR3BHTR3A
SCHEMBL29272694 0.77 GPR84 (0.74) ALDH1A1ATMGPR84KDM4EGABRA1
Hydrochloric Acid SCHEMBL29435427 0.77 GPR84 (0.74) ALDH1A1ATMGPR84KDM4EGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0922042-A1 NOVEL PIPERAZINE CONTAINING COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1999-06-16 EP disclosed
WO-1998006715-A1 NOVEL PIPERAZINE CONTAINING COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1998-02-19 WO disclosed