SCHEMBL8307482

SCHEMBL8307482

C=CCc1c(-c2cc(=O)c3c(O)c(CC=C)c(O)cc3o2)ccc(OC)c1O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 2/20 0.56
PTGES O14684 1/20 0.51
ALOX5 P09917 1/20 0.51
ABCG2 Q9UNQ0 1/20 0.49
HDAC6 Q9UBN7 1/20 0.48
PTPN1 P18031 1/20 0.47
CYP1B1 Q16678 3/20 0.46
FLT3 P36888 3/20 0.46
CYP1A1 P04798 2/20 0.46
HSD17B2 P37059 1/20 0.46
TAS2R31 P59538 1/20 0.46
AURKA O14965 1/20 0.46
KDR P35968 1/20 0.46
AURKB Q96GD4 1/20 0.46
CYP1A2 P05177 1/20 0.44
OPRD1 P41143 1/20 0.44
MMP3 P08254 1/20 0.44
MMP9 P14780 1/20 0.44
HPGD P15428 1/20 0.44
MEN1 O00255 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8309333 0.89 CYP1B1 (0.57) AKT1HDAC6PTPN1CYP1B1FLT3
SCHEMBL8304148 0.85 DYRK1A (0.49) AKT1CYP1B1CYP1A1CYP1A2HPGD
SCHEMBL8305265 0.85 CYP1B1 (0.65) AKT1PTGESALOX5ABCG2HDAC6
SCHEMBL8308046 0.84 MAOB (0.52) ABCG2HDAC6CYP1B1FLT3CYP1A1
SCHEMBL30598448 0.84 ALDH1A1 (0.43) PTPN1CYP1B1CYP1A1CYP1A2HPGD
SCHEMBL4574807 0.84 ALDH1A1 (0.43) PTPN1CYP1B1CYP1A1CYP1A2HPGD
SCHEMBL8308179 0.84 HDAC6 (0.51) AKT1PTGESALOX5HDAC6CYP1B1
SCHEMBL8305275 0.83 AKT1 (0.42) AKT1PTGESALOX5ABCG2HDAC6
SCHEMBL8429592 0.82 XDH (0.52) ABCG2HDAC6CYP1B1FLT3CYP1A1
SCHEMBL8305036 0.81 MAPT (0.59) ABCG2HDAC6CYP1B1CYP1A1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709383-B1 Diosmetin derivatives, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1999-12-15 EP disclosed
US-5629339-A CHRONIC VENOUS INSUFFICIENCY ADIR ET COMPAGNIE (FR) 1997-05-13 US disclosed
EP-0709383-A1 Diosmetin derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-05-01 EP disclosed