SCHEMBL8307770

SCHEMBL8307770

CCc1cccc2c1N(C(=N)Nc1cccc3ccccc13)CC2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 11/20 0.49
TAAR1 Q96RJ0 2/20 0.49
MAPT P10636 2/20 0.49
ALDH1A1 P00352 5/20 0.46
HSD17B10 Q99714 5/20 0.46
CYP2C19 P33261 1/20 0.46
POLB P06746 1/20 0.45
CHRM2 P08172 1/20 0.43
CHRM4 P08173 1/20 0.43
CHRM1 P11229 1/20 0.43
CHRM3 P20309 1/20 0.43
HPGD P15428 1/20 0.43
EPHX1 P07099 1/20 0.42
TSHR P16473 1/20 0.41
GAA P10253 1/20 0.40
HTR1A P08908 1/20 0.40
DRD2 P14416 1/20 0.40
USP2 O75604 1/20 0.40
LMNA P02545 1/20 0.40
ALOX15 P16050 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6768941 0.78 SIGMAR1 (0.55) KDM4ETAAR1MAPTALDH1A1HSD17B10
SCHEMBL8440692 0.78 MAPT (0.74) TAAR1MAPTALDH1A1POLBTSHR
SCHEMBL6768523 0.77 KDM4E (0.50) KDM4ETAAR1MAPTALDH1A1HSD17B10
SCHEMBL6720679 0.72 ALDH1A1 (0.55) KDM4EMAPTALDH1A1HSD17B10CYP2C19
SCHEMBL8300580 0.71 MAPT (0.49) KDM4ETAAR1MAPTALDH1A1CYP2C19
SCHEMBL8330596 0.70 GAA (0.48) KDM4ETAAR1MAPTALDH1A1HSD17B10
Hydrochloric Acid SCHEMBL6929672 0.70 CHRM2 (0.58) KDM4ETAAR1MAPTALDH1A1CHRM2
SCHEMBL8335230 0.70 NOTUM (0.48) KDM4ETAAR1MAPTALDH1A1HSD17B10
SCHEMBL7103078 0.67 ALDH1A1 (0.53) KDM4EMAPTALDH1A1HSD17B10CYP2C19
Hydrochloric Acid SCHEMBL6770312 0.66 KDM4E (0.45) KDM4ETAAR1MAPTALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0925300-A1 PHARMACEUTICALLY ACTIVE COMPOUNDS AND METHODS OF USE CAMBRIDGE NEUROSCIENCE, INC. (US) 1999-06-30 EP disclosed
EP-0925300-A4 1999-06-30 EP disclosed
WO-1997030054-A1 PHARMACEUTICALLY ACTIVE COMPOUNDS AND METHODS OF USE CAMBRIDGE NEUROSCIENCE, INC. (US) 1997-08-21 WO disclosed